Design and synthesis of somatostatin analogs with topographical properties that lead to highly potent and specific .mu. opioid receptor antagonists with greatly reduced binding at somatostatin receptors

1988 ◽  
Vol 31 (11) ◽  
pp. 2170-2177 ◽  
Author(s):  
Wieslaw Kazmierski ◽  
William S. Wire ◽  
George K. Lui ◽  
Richard J. Knapp ◽  
Jennifer E. Shook ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Somatostatin Receptors ◽  
Somatostatin Analogs ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Design And Synthesis ◽  
Opioid Receptor Antagonists

scholarly journals Naloxegol: First oral peripherally acting mu opioid receptor antagonists for opioid-induced constipation

2015 ◽  
Vol 6 (3) ◽  
pp. 188 ◽  
Author(s):  
Tejus Anantharamu ◽  
Sushil Sharma ◽  
AjayKumar Gupta ◽  
Navdeep Dahiya ◽  
DickB Singh Brashier ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Opioid Receptor Antagonists

PERIPHERALLY ACTING MU-OPIOID RECEPTOR ANTAGONISTS

2017 ◽  
Vol 40 (6) ◽  
pp. 517-522
Author(s):  
Stephanie Martinez-Cox ◽  
Karla Espinosa ◽  
Chad Friece ◽  
Anita Rahman
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Opioid Receptor Antagonists

Peripherally Acting Mu-Opioid Receptor Antagonists and Postoperative Ileus: Mechanisms of Action and Clinical Applicability

2009 ◽  
Vol 108 (6) ◽  
pp. 1811-1822 ◽  
Author(s):  
Eugene R. Viscusi ◽  
Tong J. Gan ◽  
John B. Leslie ◽  
Joseph F. Foss ◽  
Mark D. Talon ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Postoperative Ileus ◽  
Mechanisms Of Action ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Clinical Applicability ◽  
Opioid Receptor Antagonists

ChemInform Abstract: Mu Opioid Receptor Antagonists: Recent Developments

ChemInform ◽  
2008 ◽  
Vol 39 (6) ◽  
Author(s):  
Allan J. Goodman ◽  
Bertrand Le Bourdonnec ◽  
Roland E. Dolle
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Opioid Receptor Antagonists ◽  
Recent Developments

Mu Opioid Receptor Antagonists: Recent Developments

ChemMedChem ◽  
2007 ◽  
Vol 2 (11) ◽  
pp. 1552-1570 ◽  
Author(s):  
Allan J. Goodman ◽  
Bertrand Le Bourdonnec ◽  
Roland E. Dolle
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
Receptor Antagonists ◽  
Mu Opioid ◽  
Opioid Receptor Antagonists ◽  
Recent Developments
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