Molecular structures, conformational analysis, and preferential modes of binding of 3-aroyl-2-arylbenzo[b]thiophene estrogen receptor ligands: LY117018 and aryl azide photoaffinity labeling analogs

1993 ◽  
Vol 36 (24) ◽  
pp. 3910-3922 ◽  
Author(s):  
Philip R. Kym ◽  
Gregory M. Anstead ◽  
Kevin G. Pinney ◽  
Scott R. Wilson ◽  
John A. Katzenellenbogen
Keyword(s):  
Estrogen Receptor ◽  
Conformational Analysis ◽  
Photoaffinity Labeling ◽  
Molecular Structures ◽  
Receptor Ligands ◽  
Aryl Azide ◽  
Estrogen Receptor Ligands

Conformational Analysis of Bivalent Estrogen Receptor Ligands: From Intramolecular to Intermolecular Binding

ChemBioChem ◽  
2011 ◽  
Vol 12 (17) ◽  
pp. 2587-2598 ◽  
Author(s):  
Min Shan ◽  
Alexander Bujotzek ◽  
Frank Abendroth ◽  
Anja Wellner ◽  
Ronald Gust ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Conformational Analysis ◽  
Receptor Ligands ◽  
Estrogen Receptor Ligands

scholarly journals Identification of pathway-selective estrogen receptor ligands that inhibit NF- B transcriptional activity

2005 ◽  
Vol 102 (7) ◽  
pp. 2543-2548 ◽  
Author(s):  
C. C. Chadwick ◽  
S. Chippari ◽  
E. Matelan ◽  
L. Borges-Marcucci ◽  
A. M. Eckert ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Transcriptional Activity ◽  
Receptor Ligands ◽  
Estrogen Receptor Ligands

Estrogen Receptor Ligands. Part 15: Synthesis of Benzothiopyran-based Selective Estrogen Receptor Alpha Modulators (SERAM)

Heterocycles ◽  
2006 ◽  
Vol 67 (1) ◽  
pp. 79 ◽  
Author(s):  
Seongkon Kim ◽  
Frank DiNinno ◽  
Elizabeth T. Birzin ◽  
Wanda Chan ◽  
Yi Tien Yang ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Estrogen Receptor Alpha ◽  
Receptor Ligands ◽  
Receptor Alpha ◽  
Estrogen Receptor Ligands
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