Structure-activity relationships in the trans-hexahydroindolo[4,3-ab]phenanthridine ("benzergoline") series. 2. Resolution, absolute configuration, and dopaminergic activity of the selective D1 agonist CY 208-243 and its implication for an "extended rotamer-based dopamine receptor model"

1993 ◽  
Vol 36 (8) ◽  
pp. 977-984 ◽  
Author(s):  
Max P. Seiler ◽  
Philipp Floersheim ◽  
Rudolf Markstein ◽  
Armin Widmer
Keyword(s):  
Dopamine Receptor ◽  
Absolute Configuration ◽  
Receptor Model ◽  
Dopaminergic Activity ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
D1 Agonist

scholarly journals Synthesis and Structure-Activity Relationships of New (5R,8S,10R)-Ergoline Derivatives with Antihypertensive or Dopaminergic Activity.

1994 ◽  
Vol 42 (10) ◽  
pp. 2042-2048 ◽  
Author(s):  
Sachio OHNO ◽  
Masayuki KOUMORI ◽  
Yuko ADACHI(nee EBIHARA) ◽  
Kiyoshi MIZUKOSHI ◽  
Mitsuaki NAGASAKA ◽  
...  
Keyword(s):  
Dopaminergic Activity ◽  
Structure Activity Relationships ◽  
Structure Activity

scholarly journals Synthesis and Structure-Activity Relationships of New (5R,8R,10R)-Ergoline Derivatives with Antihypertensive or Dopaminergic Activity.

1994 ◽  
Vol 42 (7) ◽  
pp. 1463-1473 ◽  
Author(s):  
Sachio OHNO ◽  
Yuko ADACHI ◽  
Masayuki KOUMORI ◽  
Kiyoshi MIZUKOSHI ◽  
Mitsuaki NAGASAKA ◽  
...  
Keyword(s):  
Dopaminergic Activity ◽  
Structure Activity Relationships ◽  
Structure Activity

Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists

2005 ◽  
Vol 13 (19) ◽  
pp. 5647-5657 ◽  
Author(s):  
Simone Lorenzi ◽  
Marco Mor ◽  
Fabrizio Bordi ◽  
Silvia Rivara ◽  
Mirko Rivara ◽  
...  
Keyword(s):  
Receptor Model ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Synthesis and dopaminergic activity of some 3-(1,2,3,6-tetrahydro-1-pyridylalkyl)indoles. A novel conformational model to explain structure-activity relationships

1992 ◽  
Vol 35 (22) ◽  
pp. 4020-4026 ◽  
Author(s):  
Henning Boettcher ◽  
Gerhard Barnickel ◽  
Hans Heinrich Hausberg ◽  
Anton F. Haase ◽  
Christoph A. Seyfried ◽  
...  
Keyword(s):  
Dopaminergic Activity ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Conformational Model
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