Probing Microbiome Genotoxicity: A Stable Colibactin Provides Insight into Structure–Activity Relationships and Facilitates Mechanism of Action Studies

Journal of the American Chemical Society ◽

10.1021/jacs.1c07559 ◽

2021 ◽

Author(s):

Kevin M. Wernke ◽

Alina Tirla ◽

Mengzhao Xue ◽

Yulia V. Surovtseva ◽

Fabian S. Menges ◽

...

Keyword(s):

Mechanism Of Action ◽

Structure Activity Relationships ◽

Structure Activity ◽

Insight Into

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1,3,4-Oxadiazole-containing Hybrids as Potential Anticancer Agents: Recent Developments, Mechanism of Action and Structure-Activity Relationships

Journal of Saudi Chemical Society ◽

10.1016/j.jscs.2021.101284 ◽

2021 ◽

pp. 101284

Author(s):

Swarnagowri Nayak ◽

Santosh L. Gaonkar ◽

Ebraheem Abdu Musad ◽

Abdullah Mohammed AL. Dawsar

Keyword(s):

Mechanism Of Action ◽

Anticancer Agents ◽

Structure Activity Relationships ◽

Structure Activity ◽

Recent Developments

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Mechanistic Insight into Aerobic Alcohol Oxidation Using NOx–Nitroxide Catalysis Based on Catalyst Structure–Activity Relationships

The Journal of Organic Chemistry ◽

10.1021/jo501862k ◽

2014 ◽

Vol 79 (21) ◽

pp. 10256-10268 ◽

Cited By ~ 26

Author(s):

Masatoshi Shibuya ◽

Shota Nagasawa ◽

Yuji Osada ◽

Yoshiharu Iwabuchi

Keyword(s):

Alcohol Oxidation ◽

Catalyst Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Mechanistic Insight ◽

Insight Into

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Structure-activity relationships forPimephalesandTetrahymena: A mechanism of action approach

Environmental Toxicology and Chemistry ◽

10.1002/etc.5620160629 ◽

1997 ◽

Vol 16 (6) ◽

pp. 1311-1317 ◽

Cited By ~ 6

Author(s):

Anna P. Bearden ◽

T. Wayne Schultz

Keyword(s):

Mechanism Of Action ◽

Structure Activity Relationships ◽

Structure Activity

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Novel human umbilical vein endothelial cells (HUVEC)-apoptosis inhibitory phytosterol analogues: Insight into their structure-activity relationships

Archives of Pharmacal Research ◽

10.1007/s12272-012-0308-3 ◽

2012 ◽

Vol 35 (3) ◽

pp. 455-460 ◽

Cited By ~ 4

Author(s):

Sujin Lee ◽

Sony Marharjan ◽

Jong-Wha Jung ◽

Nam-Jung Kim ◽

Kyeojin Kim ◽

...

Keyword(s):

Endothelial Cells ◽

Umbilical Vein ◽

Human Umbilical Vein ◽

Structure Activity Relationships ◽

Structure Activity ◽

Umbilical Vein Endothelial Cells ◽

Insight Into

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Norepinephrine alkaloids as antiplasmodial agents: Synthesis of syncarpamide and insight into the structure-activity relationships of its analogues as antiplasmodial agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2017.07.052 ◽

2017 ◽

Vol 138 ◽

pp. 1089-1105 ◽

Cited By ~ 8

Author(s):

Eswar K. Aratikatla ◽

Tushar R. Valkute ◽

Sunil K. Puri ◽

Kumkum Srivastava ◽

Asish K. Bhattacharya

Keyword(s):

Structure Activity Relationships ◽

Structure Activity ◽

Insight Into

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Structure-Activity Relationships and Mechanism of Action of Macrolides Derived from Erythromycin as Antibacterial Agents

Current Topics in Medicinal Chemistry ◽

10.2174/15680266113136660223 ◽

2013 ◽

Vol 13 (24) ◽

pp. 3131-3164 ◽

Cited By ~ 25

Author(s):

Jian-Hua Liang ◽

Xu Han

Keyword(s):

Mechanism Of Action ◽

Antibacterial Agents ◽

Structure Activity Relationships ◽

Structure Activity

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Faculty Opinions recommendation of The solution structure of Bacillus anthracis dihydrofolate reductase yields insight into the analysis of structure-activity relationships for novel inhibitors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1159058.619347 ◽

2009 ◽

Author(s):

Vivian Cody

Keyword(s):

Bacillus Anthracis ◽

Dihydrofolate Reductase ◽

Solution Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Insight Into

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STRUCTURE–ACTIVITY RELATIONSHIPS FOR PIMEPHALES AND TETRAHYMENA: A MECHANISM OF ACTION APPROACH

Environmental Toxicology and Chemistry ◽

10.1897/1551-5028(1997)016<1311:sarfpa>2.3.co;2 ◽

1997 ◽

Vol 16 (6) ◽

pp. 1311 ◽

Cited By ~ 5

Author(s):

Anna P. Bearden ◽

T. Wayne Schultz

Keyword(s):

Mechanism Of Action ◽

Structure Activity Relationships ◽

Structure Activity

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Structure–activity relationships of 4-N-substituted ferroquine analogues: Time to re-evaluate the mechanism of action of ferroquine

Journal of Organometallic Chemistry ◽

10.1016/j.jorganchem.2008.09.033 ◽

2009 ◽

Vol 694 (6) ◽

pp. 845-854 ◽

Cited By ~ 42

Author(s):

Christophe Biot ◽

Natascha Chavain ◽

Faustine Dubar ◽

Bruno Pradines ◽

Xavier Trivelli ◽

...

Keyword(s):

Mechanism Of Action ◽

Structure Activity Relationships ◽

Structure Activity

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Structure–Activity Relationships and Mechanism of Action of Small Molecule Smoothened Modulators Discovered by High-Throughput Screening and Rational Design

Topics in Medicinal Chemistry - The Smoothened Receptor in Cancer and Regenerative Medicine ◽

10.1007/7355_2014_61 ◽

2014 ◽

pp. 43-107 ◽

Cited By ~ 5

Author(s):

Fabrizio Manetti ◽

Maurizio Taddei ◽

Elena Petricci

Keyword(s):

Small Molecule ◽

High Throughput ◽

Mechanism Of Action ◽

High Throughput Screening ◽

Rational Design ◽

Structure Activity Relationships ◽

Structure Activity

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