Microwave-Assisted Tandem Cross Metathesis Intramolecular Aza-Michael Reaction:  An Easy Entry to Cyclic β-Amino Carbonyl Derivatives

2007 ◽  
Vol 129 (21) ◽  
pp. 6700-6701 ◽  
Author(s):  
Santos Fustero ◽  
Diego Jiménez ◽  
María Sánchez-Roselló ◽  
Carlos del Pozo
Keyword(s):  
Michael Reaction ◽  
Microwave Assisted ◽  
Cross Metathesis ◽  
Carbonyl Derivatives

scholarly journals Microwave-assisted telescoped cross metathesis-ring closing aza-Michael reaction sequence: step-economical access to nicotine–lobeline hybrid analogues

RSC Advances ◽  
2015 ◽  
Vol 5 (117) ◽  
pp. 96720-96724 ◽  
Author(s):  
E. Drège ◽  
J. Oko ◽  
P.-E. Venot ◽  
N. Gigant ◽  
D. Joseph
Keyword(s):  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Michael Addition ◽  
Michael Reaction ◽  
Receptor Ligands ◽  
Reaction Sequence ◽  
Nicotinic Acetylcholine ◽  
Microwave Assisted ◽  
Cross Metathesis

Step-economical access to nicotinic acetylcholine receptor ligands hybrids through an efficient telescoped cross-metathesis/cyclizing aza-Michael addition involving N-heteroaromatic olefinic derivatives.

Synthesis of Substituted β‐Functionalised Styrenes by Microwave‐Assisted Olefin Cross‐Metathesis and Scalable Synthesis of Apremilast

ChemCatChem ◽  
2019 ◽  
Vol 11 (23) ◽  
pp. 5808-5813 ◽  
Author(s):  
Anupam Jana ◽  
Grzegorz Krzysztof Zieliński ◽  
Sylwia Czarnocka‐Śniadała ◽  
Krzysztof Grudzień ◽  
Dominika Podwysocka ◽  
...  
Keyword(s):  
Microwave Assisted ◽  
Cross Metathesis ◽  
Scalable Synthesis

ChemInform Abstract: Microwave-Assisted Tandem Organocatalytic Peptide-Coupling Intramolecular aza-Michael Reaction: α,β-Unsaturated N-Acyl Pyrazoles as Michael Acceptors.

ChemInform ◽  
2015 ◽  
Vol 46 (18) ◽  
pp. no-no
Author(s):  
Maria Sanchez-Rosello ◽  
Cristina Mulet ◽  
Marta Guerola ◽  
Carlos del Pozo ◽  
Santos Fustero
Keyword(s):  
Michael Reaction ◽  
Peptide Coupling ◽  
Microwave Assisted ◽  
Michael Acceptors

An Novel Synthesis Route of γ-Nitro-β-Aryl-α-Methylene Arone: Microwave-Assisted Michael Reaction of Phosphorus Ylides to Nitroolefins

2013 ◽  
Vol 291-294 ◽  
pp. 730-733
Author(s):  
Yi Si Yang ◽  
Yan Zhang
Keyword(s):  
Microwave Irradiation ◽  
Michael Reaction ◽  
Phosphorus Ylides ◽  
Subsequent Reaction ◽  
Microwave Assisted ◽  
Synthesis Route ◽  
Novel Synthesis ◽  
Michael Type Addition ◽  
Microwave Time ◽  
First Time

Michael-type addition of stabilized phosphorus ylides to nitroolefins was accomplished under microwave irradiation for the first time. Its subsequent reaction with formaldehyde provides γ-nitro-β-aryl-α-methylene arone. The solvents, microwave time and power were screened, the best yield was got(up to 62% ).

A New Tandem Cross Metathesis-Intramolecular Aza-Michael Reaction for the Synthesis of α,α-Difluorinated Lactams

Synthesis ◽  
2012 ◽  
Vol 44 (12) ◽  
pp. 1863-1873 ◽  
Author(s):  
Santos Fustero ◽  
Carlos del Pozo ◽  
Claribel Báez ◽  
María Sánchez-Roselló ◽  
Amparo Asensio ◽  
...  
Keyword(s):  
Michael Reaction ◽  
Cross Metathesis

Total Synthesis of Cystothiazole A by Microwave-Assisted Olefin Cross-Metathesis

2008 ◽  
Vol 2008 (16) ◽  
pp. 2701-2704 ◽  
Author(s):  
Julian Gebauer ◽  
Stellios Arseniyadis ◽  
Janine Cossy
Keyword(s):  
Total Synthesis ◽  
Microwave Assisted ◽  
Cross Metathesis
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