New Transient Receptor Potential Vanilloid Subfamily Member 1 Positron Emission Tomography Radioligands: Synthesis, Radiolabeling, and Preclinical Evaluation

Daisy van Veghel; Jan Cleynhens; Larry V. Pearce; Ian A. DeAndrea-Lazarus; Peter M. Blumberg; Koen Van Laere; Alfons Verbruggen; Guy Bormans

doi:10.1021/cn300233v

New Transient Receptor Potential Vanilloid Subfamily Member 1 Positron Emission Tomography Radioligands: Synthesis, Radiolabeling, and Preclinical Evaluation

ACS Chemical Neuroscience ◽

10.1021/cn300233v ◽

2013 ◽

Vol 4 (4) ◽

pp. 624-634 ◽

Cited By ~ 6

Author(s):

Daisy van Veghel ◽

Jan Cleynhens ◽

Larry V. Pearce ◽

Ian A. DeAndrea-Lazarus ◽

Peter M. Blumberg ◽

...

Keyword(s):

Positron Emission Tomography ◽

Transient Receptor Potential ◽

Receptor Potential ◽

Emission Tomography ◽

Transient Receptor Potential Vanilloid ◽

Preclinical Evaluation ◽

Subfamily Member ◽

Positron Emission ◽

Transient Receptor

Download Full-text

Sa1216 IN PATIENTS WITH HEARTBURN, SUPERFICIAL MUCOSAL AFFERENT NERVES EXPRESS TRANSIENT RECEPTOR POTENTIAL VANILLOID SUBFAMILY MEMBER-1 (TRPV1)

Gastroenterology ◽

10.1016/s0016-5085(20)31488-8 ◽

2020 ◽

Vol 158 (6) ◽

pp. S-315-S-316

Author(s):

Ahsen Ustaoglu ◽

Philip J. Woodland ◽

Madusha Peiris ◽

Chung Lee ◽

Kornilia Nikaki ◽

...

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Subfamily Member ◽

Afferent Nerves ◽

Transient Receptor

Download Full-text

Synthesis and vasodilator effects of rutaecarpine analogues which might be involved transient receptor potential vanilloid subfamily, member 1 (TRPV1)

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.02.015 ◽

2009 ◽

Vol 17 (6) ◽

pp. 2351-2359 ◽

Cited By ~ 59

Author(s):

Zhuo Chen ◽

Gaoyun Hu ◽

Dai Li ◽

Jun Chen ◽

Yuanjian Li ◽

...

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Subfamily Member ◽

Transient Receptor

Download Full-text

[ 11 C]BCTC: Radiosynthesis and in vivo binding to transient receptor potential vanilloid subfamily member 1 (TRPV1) receptor in the mouse trigeminal nerve

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2017.08.061 ◽

2017 ◽

Vol 27 (19) ◽

pp. 4521-4524

Author(s):

Katsushi Kumata ◽

Joji Yui ◽

Yiding Zhang ◽

Yusuke Kurihara ◽

Masanao Ogawa ◽

...

Keyword(s):

Trigeminal Nerve ◽

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Trpv1 Receptor ◽

In Vivo Binding ◽

Subfamily Member ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of Transient receptor potential vanilloid 1 is required for intrinsic osmoreception in organum vasculosum lamina terminalis neurons and for normal thirst responses to systemic hyperosmolality.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1047186.497222 ◽

2006 ◽

Author(s):

Alastair Ferguson

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Lamina Terminalis ◽

Organum Vasculosum Lamina Terminalis ◽

Organum Vasculosum ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of Transient receptor potential vanilloid 1 is required for intrinsic osmoreception in organum vasculosum lamina terminalis neurons and for normal thirst responses to systemic hyperosmolality.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1047186.497108 ◽

2006 ◽

Author(s):

Bernd Nilius

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Lamina Terminalis ◽

Organum Vasculosum Lamina Terminalis ◽

Organum Vasculosum ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of Somatostatin modulates the transient receptor potential vanilloid 1 (TRPV1) ion channel.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1052995.504951 ◽

2006 ◽

Author(s):

Marcos Milla

Keyword(s):

Ion Channel ◽

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of A specific subset of transient receptor potential vanilloid-type channel subunits in Caenorhabditis elegans endocrine cells function as mixed heteromers to promote neurotransmitter release.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1063770.516694 ◽

2007 ◽

Author(s):

Oliver Hobert

Keyword(s):

Caenorhabditis Elegans ◽

Neurotransmitter Release ◽

Endocrine Cells ◽

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Specific Subset ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of Activation of urothelial transient receptor potential vanilloid 4 by 4alpha-phorbol 12,13-didecanoate contributes to altered bladder reflexes in the rat.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1100237.558108 ◽

2008 ◽

Author(s):

Rodolfo Testa

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of Design and synthesis of peripherally restricted transient receptor potential vanilloid 1 (TRPV1) antagonists.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1108621.564704 ◽

2008 ◽

Author(s):

Rodolfo Testa

Keyword(s):

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Design And Synthesis ◽

Transient Receptor

Download Full-text

Faculty Opinions recommendation of The mechanosensitivity of mouse colon afferent fibers and their sensitization by inflammatory mediators require transient receptor potential vanilloid 1 and acid-sensing ion channel 3.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.7001.464490 ◽

2006 ◽

Author(s):

Gyongyi Horvath

Keyword(s):

Ion Channel ◽

Inflammatory Mediators ◽

Transient Receptor Potential ◽

Receptor Potential ◽

Transient Receptor Potential Vanilloid ◽

Mouse Colon ◽

Afferent Fibers ◽

Transient Receptor

Download Full-text