Structure—Activity Study and Conformational Analysis of RH—5992, the First Commercialized Nonsteroidal Ecdysone Agonist

A study of the structure–activity relationship of GABAA–benzodiazepine receptor bivalent ligands by conformational analysis with low temperature NMR and X-ray analysis

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.08.072 ◽

2008 ◽

Vol 16 (19) ◽

pp. 8853-8862 ◽

Cited By ~ 6

Author(s):

Dongmei Han ◽

F. Holger Försterling ◽

Xiaoyan Li ◽

Jeffrey R. Deschamps ◽

Damon Parrish ◽

...

Keyword(s):

Low Temperature ◽

Conformational Analysis ◽

Benzodiazepine Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Bivalent Ligands ◽

X Ray ◽

Structure Activity ◽

Relationship Of

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ChemInform Abstract: CAMBRIDGE DATA FILE IN ORGANIC CHEMISTRY. APPLICATIONS TO TRANSITION-STATE STRUCTURE, CONFORMATIONAL ANALYSIS, AND STRUCTURE/ACTIVITY STUDIES

Chemischer Informationsdienst ◽

10.1002/chin.198023088 ◽

1980 ◽

Vol 11 (23) ◽

Author(s):

S. R. WILSON ◽

J. C. HUFFMAN

Keyword(s):

Organic Chemistry ◽

Transition State ◽

Conformational Analysis ◽

Data File ◽

State Structure ◽

Transition State Structure ◽

Structure Activity

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Dienic analogs of (Z)-5-decenyl acetate, a pheromone component of the turnip moth, Agrotis segetum: Synthesis, conformational analysis and structure-activity relationships

Bioorganic Chemistry ◽

10.1016/0045-2068(87)90036-8 ◽

1987 ◽

Vol 15 (4) ◽

pp. 409-422 ◽

Cited By ~ 25

Author(s):

Marie Bengtsson ◽

Tommy Liljefors ◽

Bill S. Hansson

Keyword(s):

Conformational Analysis ◽

Pheromone Component ◽

Agrotis Segetum ◽

Structure Activity Relationships ◽

Structure Activity ◽

Turnip Moth

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Structure–activity relationship and conformational analysis of monoglycosylceramides on the syngeneic mixed leukocyte reaction

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(98)00112-6 ◽

1998 ◽

Vol 6 (10) ◽

pp. 1905-1910 ◽

Cited By ~ 14

Author(s):

Hiroshi Iijima ◽

Kaname Kimura ◽

Teruyuki Sakai ◽

Akira Uchimura ◽

Toshiyuki Shimizu ◽

...

Keyword(s):

Conformational Analysis ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Mixed Leukocyte Reaction ◽

Structure Activity

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ChemInform Abstract: Benzoxazines. Part 2. Synthesis, Conformational Analysis, and Structure-Activity Relationships of 3,4-Dihydro-2H-1,4-benzoxazine-8- carboxamide Derivatives as Potent and Long-Acting Serotonin-3 (5-HT3) Receptor Antagonists.

ChemInform ◽

10.1002/chin.199721050 ◽

2010 ◽

Vol 28 (21) ◽

pp. no-no

Author(s):

T. KUROITA ◽

N. MARUBAYASHI ◽

M. SANO ◽

K. KANZAKI ◽

K. INABA ◽

...

Keyword(s):

Conformational Analysis ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity ◽

Long Acting

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Three-Dimensional Structure-Activity Relationship Analysis between Motilin and Motilide Using Conformational Analysis and a Novel Molecular Superposing Method.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.48.1835 ◽

2000 ◽

Vol 48 (11) ◽

pp. 1835-1837 ◽

Cited By ~ 2

Author(s):

Hiroaki GOUDA ◽

Toshiaki SUNAZUKA ◽

Satoshi OMURA ◽

Shuichi HIRONO

Keyword(s):

Conformational Analysis ◽

Three Dimensional ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Dimensional Structure ◽

Three Dimensional Structure ◽

Relationship Analysis ◽

Structure Activity

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Isovanillyl sweeteners. Synthesis, conformational analysis, and structure–activity relationship of some sweet oxygen heterocycles

Journal of the Chemical Society Perkin Transactions 2 ◽

10.1039/p29910001399 ◽

1991 ◽

pp. 1399-1406 ◽

Cited By ~ 15

Author(s):

Anna Arnoldi ◽

Angela Bassoli ◽

Lucio Merlini ◽

Enzio Ragg

Keyword(s):

Conformational Analysis ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Oxygen Heterocycles ◽

Relationship Of

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Conformational analysis of podophyllotoxin and its congeners. Structure-activity relationship in microtubule assembly

Journal of Medicinal Chemistry ◽

10.1021/jm00189a001 ◽

1979 ◽

Vol 22 (3) ◽

pp. 215-221 ◽

Cited By ~ 87

Author(s):

C. Fred Brewer ◽

John D. Loike ◽

Susan B. Horwitz ◽

Himan Sternlicht ◽

Walter J. Gensler

Keyword(s):

Conformational Analysis ◽

Structure Activity Relationship ◽

Microtubule Assembly ◽

Activity Relationship ◽

Structure Activity

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Statistical analysis and shape recognition: Applications to MD simulations, conformational analysis and structure-activity relationships

Trends in QSAR and Molecular Modelling 92 ◽

10.1007/978-94-011-1472-1_33 ◽

1993 ◽

pp. 216-219 ◽

Cited By ~ 3

Author(s):

Gérard Grassy ◽

Roger Lahana

Keyword(s):

Statistical Analysis ◽

Conformational Analysis ◽

Shape Recognition ◽

Md Simulations ◽

Structure Activity Relationships ◽

Structure Activity

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SYNTHESIS AND BIOLOGICAL ACTIVITY OF CYCLIC ADP-CARBOCYCLIC-RIBOSE ANALOGS: STRUCTURE-ACTIVITY RELATIONSHIP AND CONFORMATIONAL ANALYSIS OF N-1-CARBOCYCLIC-RIBOSE MOIETY

Nucleosides Nucleotides & Nucleic Acids ◽

10.1081/ncn-200060167 ◽

2005 ◽

Vol 24 (5-7) ◽

pp. 655-658 ◽

Cited By ~ 1

Author(s):

Takashi Kudoh ◽

Masayoshi Fukuoka ◽

Satoshi Shuto ◽

Akira Matsuda

Keyword(s):

Biological Activity ◽

Conformational Analysis ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Ribose Moiety

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