scholarly journals Molecular Characterization of Agonists That Bind to an Insect GABA Receptor

Biochemistry ◽  
2010 ◽  
Vol 49 (13) ◽  
pp. 2897-2902 ◽  
Author(s):  
Ian McGonigle ◽  
Sarah C. R. Lummis
Keyword(s):  
Molecular Characterization ◽  
Gaba Receptor

scholarly journals A molecular characterization of the agonist binding site of a nematode cys-loop GABA receptor

2015 ◽  
Vol 172 (15) ◽  
pp. 3737-3747 ◽  
Author(s):  
Mark D Kaji ◽  
Ariel Kwaka ◽  
Micah K Callanan ◽  
Humza Nusrat ◽  
Jean-Paul Desaulniers ◽  
...  
Keyword(s):  
Binding Site ◽  
Molecular Characterization ◽  
Gaba Receptor ◽  
Agonist Binding

Molecular Characterization of Avermectin that Bind to Rdl β5 GABA Receptors of House Fly

2013 ◽  
Vol 699 ◽  
pp. 753-758 ◽  
Author(s):  
Ming Hao ◽  
Qiang Wang ◽  
Qing Qing Ma ◽  
Jin Long Zhao ◽  
Wan Guo Hou ◽  
...  
Keyword(s):  
Hydrogen Bond ◽  
Free Energy ◽  
Molecular Characterization ◽  
Hydrophobic Interaction ◽  
Gaba Receptors ◽  
Gaba Receptor ◽  
Binding Free Energy ◽  
House Fly ◽  
Before And After

The interaction between Rdlβ5 GABA receptors of house fly before and after mutation and AVM was considered as the reason that AVM cause the insect death and investigated with Sybylx1.1 software. The docking results showed that the hydrogen bond and hydrophobic interaction played an important role among the complexes of Rdlβ5 GABA receptor and avermectin. Hydrogen bond of 2.217 Å formed between B/Ser58 of GABA receptor and atom O42 of avermectin before mutation, 1.953 Å hydrogen bond formed between A/Gln6 of GABA receptor and hydroxyl (C7) of avermectin after mutation. In addition, our results indicated that the binding free energy (ΔE) of AVM and GABA receptors increased 3.59 kcal mol−1 after mutation, which was consistent with the experimental phenomenon of the insecticidal resistance to AVM.

scholarly journals Molecular Characterization of Binding Loop E in the Nematode Cys-Loop GABA Receptor

2018 ◽  
Vol 94 (5) ◽  
pp. 1289-1297 ◽  
Author(s):  
Ariel Kwaka ◽  
Mohammad Hassan Khatami ◽  
Joshua Foster ◽  
Everett Cochrane ◽  
Sarah A. Habibi ◽  
...  
Keyword(s):  
Molecular Characterization ◽  
Gaba Receptor ◽  
Binding Loop

1446: Molecular Characterization of Cyclooxygenase-2 in a Stimulated Prostate Stroma Cells

2006 ◽  
Vol 175 (4S) ◽  
pp. 467-467
Author(s):  
Victor K. Lin ◽  
Shih-Ya Wang ◽  
Claus G. Roehrbom
Keyword(s):  
Molecular Characterization ◽  
Cyclooxygenase 2 ◽  
Prostate Stroma

Molecular characterization of lincRNAs in Down syndrome associated leukemia

2012 ◽  
Vol 224 (03) ◽  
Author(s):  
A Streltsov ◽  
S Emmrich ◽  
F Engeland ◽  
JH Klusmann
Keyword(s):  
Down Syndrome ◽  
Molecular Characterization

Molecular Characterization of Radiation-induced Glioblastoma

2018 ◽  
Author(s):  
MY Deng ◽  
D Sturm ◽  
E Pfaff ◽  
GP Balasubrama ◽  
J Schittenhelm ◽  
...  
Keyword(s):  
Molecular Characterization ◽  
Radiation Induced
Sign in / Sign up

Export Citation Format

Share Document