scholarly journals Activation of G Protein-Coupled Receptor Kinase 1 Involves Interactions between Its N-Terminal Region and Its Kinase Domain

Biochemistry ◽  
2011 ◽  
Vol 50 (11) ◽  
pp. 1940-1949 ◽  
Author(s):  
Chih-chin Huang ◽  
Tivadar Orban ◽  
Beata Jastrzebska ◽  
Krzysztof Palczewski ◽  
John J. G. Tesmer
Keyword(s):  
G Protein ◽  
Kinase Domain ◽  
Terminal Region ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
G Protein Coupled

scholarly journals Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein–Coupled Receptor Kinase 2 Inhibitors

2017 ◽  
Vol 92 (6) ◽  
pp. 707-717 ◽  
Author(s):  
Renee Bouley ◽  
Helen V. Waldschmidt ◽  
M. Claire Cato ◽  
Alessandro Cannavo ◽  
Jianliang Song ◽  
...  
Keyword(s):  
G Protein ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
Structural Determinants ◽  
G Protein Coupled

scholarly journals Generation of Highly Selective, Potent, and Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors

2021 ◽  
Author(s):  
Rachel A. Rowlands ◽  
Qiuyan Chen ◽  
Renee A. Bouley ◽  
Larisa V. Avramova ◽  
John J. G. Tesmer ◽  
...  
Keyword(s):  
G Protein ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
G Protein Coupled
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