Bicyclic Chalcones as Mitotic Inhibitors for Overcoming Androgen Receptor-Independent and Multidrug-Resistant Prostate Cancer

Yohei Saito; Atsushi Mizokami; Sayaka Maeda; Kyoko Takahashi; Kouji Izumi; Masuo Goto; Kyoko Nakagawa-Goto

doi:10.1021/acsomega.0c05822

Bicyclic Chalcones as Mitotic Inhibitors for Overcoming Androgen Receptor-Independent and Multidrug-Resistant Prostate Cancer

ACS Omega ◽

10.1021/acsomega.0c05822 ◽

2021 ◽

Vol 6 (7) ◽

pp. 4842-4849

Author(s):

Yohei Saito ◽

Atsushi Mizokami ◽

Sayaka Maeda ◽

Kyoko Takahashi ◽

Kouji Izumi ◽

...

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Multidrug Resistant ◽

Mitotic Inhibitors

Download Full-text

609: Effects of Sirna and Phytoestrogen Treatments on the Expression of Genes Regulated through the Androgen Receptor of Lncap Prostate Cancer Cells

The Journal of Urology ◽

10.1016/s0022-5347(18)37871-6 ◽

2004 ◽

Vol 171 (4S) ◽

pp. 162-162

Author(s):

Paul Thelen ◽

Michal Grzmil ◽

Iris E. Eder ◽

Barbara Spengler ◽

Peter Burfeind ◽

...

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Cancer Cells ◽

Prostate Cancer Cells ◽

Expression Of Genes

Download Full-text

The role of androgen receptor in glucose transporters expression in prostate cancer cells

Endocrine Abstracts ◽

10.1530/endoabs.37.gp.30.03 ◽

2015 ◽

Author(s):

Pedro Gonzalez-Menendez ◽

David Hevia ◽

Juan C Mayo ◽

Rosa M Sainz

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Cancer Cells ◽

Glucose Transporters ◽

Prostate Cancer Cells

Download Full-text

Modulation of androgen receptor signaling in prostate cancer cells by SUMOylation and NFκB pathways

Endocrine Abstracts ◽

10.1530/endoabs.42.il4 ◽

2016 ◽

Author(s):

Jorma J. Palvimo

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Cancer Cells ◽

Receptor Signaling ◽

Prostate Cancer Cells ◽

Androgen Receptor Signaling

Download Full-text

A genome-scale CRISPR screen reveals PRMT1 as a critical regulator of androgen receptor signaling in prostate cancer

10.26226/morressier.5f69edb69b74b699bf38c5e4 ◽

2020 ◽

Author(s):

Srinivas R. Viswanathan

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Receptor Signaling ◽

Androgen Receptor Signaling ◽

A Genome ◽

Crispr Screen ◽

Genome Scale

Download Full-text

Faculty Opinions recommendation of Systematic evaluation of genetic variation at the androgen receptor locus and risk of prostate cancer in a multiethnic cohort study.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1023470.270750 ◽

2005 ◽

Author(s):

Pui-Yan Kwok

Keyword(s):

Prostate Cancer ◽

Genetic Variation ◽

Cohort Study ◽

Androgen Receptor ◽

Systematic Evaluation ◽

Multiethnic Cohort ◽

Receptor Locus

Download Full-text

Faculty Opinions recommendation of Ligand-specific allosteric regulation of coactivator functions of androgen receptor in prostate cancer cells.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1031334.363672 ◽

2006 ◽

Author(s):

Aniko Naray-Fejes-Toth

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Cancer Cells ◽

Allosteric Regulation ◽

Prostate Cancer Cells

Download Full-text

Faculty Opinions recommendation of Reciprocal feedback regulation of PI3K and androgen receptor signaling in PTEN-deficient prostate cancer.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.10718956.11608054 ◽

2011 ◽

Author(s):

Christopher Janetopoulos

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Feedback Regulation ◽

Receptor Signaling ◽

Androgen Receptor Signaling

Download Full-text

Faculty Opinions recommendation of A hierarchical network of transcription factors governs androgen receptor-dependent prostate cancer growth.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1089669.544943 ◽

2007 ◽

Author(s):

Paul Webb

Keyword(s):

Prostate Cancer ◽

Transcription Factors ◽

Androgen Receptor ◽

Cancer Growth ◽

Hierarchical Network

Download Full-text

Faculty Opinions recommendation of Regression of castrate-recurrent prostate cancer by a small-molecule inhibitor of the amino-terminus domain of the androgen receptor.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.5059957.4994055 ◽

2010 ◽

Author(s):

Michael Weber ◽

Daniel G Gioeli

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Small Molecule ◽

Small Molecule Inhibitor ◽

Amino Terminus ◽

Recurrent Prostate Cancer ◽

Molecule Inhibitor

Download Full-text

Faculty Opinions recommendation of Resistance to CYP17A1 inhibition with abiraterone in castration-resistant prostate cancer: induction of steroidogenesis and androgen receptor splice variants.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.714997806.790402827 ◽

2012 ◽

Author(s):

Hendrik van Poppel ◽

Yuri Tolkach

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Splice Variants ◽

Castration Resistant Prostate Cancer ◽

Cancer Induction ◽

Castration Resistant ◽

Androgen Receptor Splice Variants

Download Full-text