Incorporation of Fluorine into an OBOC Peptide Library by Copper-Free Click Chemistry toward the Discovery of PET Imaging Agents

2020 ◽  
Vol 22 (3) ◽  
pp. 109-113
Author(s):  
Emily Murrell ◽  
Leonard G. Luyt
Keyword(s):  
Click Chemistry ◽  
Pet Imaging ◽  
Peptide Library ◽  
Imaging Agents

scholarly journals β-Configured clickable [18F]FDGs as novel 18F-fluoroglycosylation tools for PET

2017 ◽  
Vol 41 (18) ◽  
pp. 10231-10236 ◽  
Author(s):  
M. Elgland ◽  
P. Nordeman ◽  
T. Fyrner ◽  
G. Antoni ◽  
K. Peter R. Nilsson ◽  
...  
Keyword(s):  
Click Chemistry ◽  
Pet Imaging ◽  
Prosthetic Groups

We have developed a chemoselective 18F-fluoroglycosylation method for PET imaging that employ β-configured [18F]FDGs as prosthetic groups for 18F-labeling using CuAAC click chemistry.

Improving excretory pathways of technetium-99m SPECT imaging agents based on bioorthogonal Diels-Alder click chemistry

2019 ◽  
Vol 72-73 ◽  
pp. S65
Author(s):  
J. Walsh ◽  
L. Francesconi ◽  
V. Sanders ◽  
D. Iskhakov ◽  
B. Zeglis ◽  
...  
Keyword(s):  
Click Chemistry ◽  
Diels Alder ◽  
Spect Imaging ◽  
Imaging Agents ◽  
Technetium 99M

Synthesis and evaluation of pyridylbenzofuran, pyridylbenzothiazole and pyridylbenzoxazole derivatives as 18F-PET imaging agents for β-amyloid plaques

2012 ◽  
Vol 22 (13) ◽  
pp. 4332-4337 ◽  
Author(s):  
Britt-Marie Swahn ◽  
Johan Sandell ◽  
David Pyring ◽  
Margareta Bergh ◽  
Fredrik Jeppsson ◽  
...  
Keyword(s):  
Pet Imaging ◽  
Amyloid Plaques ◽  
Imaging Agents ◽  
Β Amyloid

Design, Synthesis, and Evaluation of a Low-Molecular-Weight 11C-Labeled Tetrazine for Pretargeted PET Imaging Applying Bioorthogonal in Vivo Click Chemistry

2016 ◽  
Vol 27 (7) ◽  
pp. 1707-1712 ◽  
Author(s):  
Christoph Denk ◽  
Dennis Svatunek ◽  
Severin Mairinger ◽  
Johann Stanek ◽  
Thomas Filip ◽  
...  
Keyword(s):  
Molecular Weight ◽  
Click Chemistry ◽  
Pet Imaging ◽  
Low Molecular Weight ◽  
Design Synthesis

Synthesis of 2-R1-2-(4-(2-fluoroethoxy)benzamido)acetate as potential PET imaging agents

2011 ◽  
Vol 21 (6) ◽  
pp. 944-951 ◽  
Author(s):  
Yong He ◽  
Jingli Xu ◽  
Hang Liu ◽  
Man Feng ◽  
Xiao Wang ◽  
...  
Keyword(s):  
Pet Imaging ◽  
Imaging Agents

scholarly journals Synthesis and evaluation of novel F-18-labeled pyrimidine derivatives: potential FAK inhibitors and PET imaging agents for cancer detection

RSC Advances ◽  
2017 ◽  
Vol 7 (36) ◽  
pp. 22388-22399 ◽  
Author(s):  
Dawei Wang ◽  
Yu Fang ◽  
Hang Wang ◽  
Xingyu Xu ◽  
Jianping Liu ◽  
...  
Keyword(s):  
Cancer Detection ◽  
Pet Imaging ◽  
Imaging Study ◽  
Imaging Agents ◽  
Post Injection ◽  
Pyrimidine Derivatives ◽  
Micropet Imaging ◽  
Tumor Bearing ◽  
Biodistribution Data

Compound [18F]-8a exhibited good in vivo biodistribution data in mice bearing S180 tumor. And the microPET imaging study of [18F]-8a in S180 tumor-bearing mice was also preformed, which illustrated that the uptake in S180 tumor at 60 min post-injection of [18F]-8a was obvious.

Sign in / Sign up

Export Citation Format

Share Document