One-Pot Construction of Indolo[2,3-b]quinoxalines through Ruthenium-Catalyzed Ortho C–H Bond Functionalization of 2-Arylquinoxalines with Sulfonyl Azides

2021 ◽  
Author(s):  
Sudip Laru ◽  
Suvam Bhattacharjee ◽  
Sumit Ghosh ◽  
Alakananda Hajra
2018 ◽  
Vol 83 (22) ◽  
pp. 14195-14202 ◽  
Author(s):  
Elina Ausekle ◽  
Peter Ehlers ◽  
Alexander Villinger ◽  
Peter Langer

Tetrahedron ◽  
2014 ◽  
Vol 70 (38) ◽  
pp. 6717-6722 ◽  
Author(s):  
Xian-chun Tan ◽  
Ying Liang ◽  
Fang-ping Bao ◽  
Heng-shan Wang ◽  
Ying-ming Pan

2019 ◽  
Vol 15 ◽  
pp. 2069-2075 ◽  
Author(s):  
Hai-Yun Huang ◽  
Haoran Li ◽  
Thierry Roisnel ◽  
Jean-François Soulé ◽  
Henri Doucet

The Pd-catalyzed C–H bond functionalization of lilolidine was investigated. The use of a palladium-diphosphine catalyst associated to acetate bases in DMA was found to promote the regioselective arylation at α-position of the nitrogen atom of lilolidine with a wide variety of aryl bromides. From these α-arylated lilolidines, a second arylation at the β-position gives the access to α,β-diarylated lilolidines containing two different aryl groups. The one pot access to α,β-diarylated lilolidines with two identical aryl groups is also possible by using a larger amount of aryl bromide. The synthesis of 5,6-dihydrodibenzo[a,c]pyrido[3,2,1-jk]carbazoles from lilolidine via three successive direct arylations is also described. Therefore, this methodology provides a straightforward access to several lilolidine derivatives from commercially available compounds via one, two or three C–H bond functionalization steps allowing to tune their biological properties.


2012 ◽  
Vol 53 (8) ◽  
pp. 942-943 ◽  
Author(s):  
Issa Yavari ◽  
Manijeh Nematpour ◽  
Majid Ghazanfarpour-Darjani

ChemInform ◽  
2012 ◽  
Vol 43 (6) ◽  
pp. no-no
Author(s):  
Hojat Veisi ◽  
Ramin Ghorbani-Vaghei ◽  
Saba Hemmati ◽  
Jafar Mahmoodi

2013 ◽  
Vol 96 (12) ◽  
pp. 2214-2217 ◽  
Author(s):  
Issa Yavari ◽  
Tahereh Damghani ◽  
Manijeh Nematpour

ChemInform ◽  
2016 ◽  
Vol 47 (14) ◽  
Author(s):  
Shanmugam Rajasekar ◽  
Dongari Yadagiri ◽  
Pazhamalai Anbarasan
Keyword(s):  
One Pot ◽  

ChemInform ◽  
2014 ◽  
Vol 45 (48) ◽  
pp. no-no
Author(s):  
Taekyu Ryu ◽  
Jiae Min ◽  
Wonseok Choi ◽  
Woo Hyung Jeon ◽  
Phil Ho Lee
Keyword(s):  
One Pot ◽  

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