Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents

Silvia Bartolucci; Michele Mari; Annalida Bedini; Giovanni Piersanti; Gilberto Spadoni

doi:10.1021/acs.joc.5b00195

Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents

The Journal of Organic Chemistry ◽

10.1021/acs.joc.5b00195 ◽

2015 ◽

Vol 80 (6) ◽

pp. 3217-3222 ◽

Cited By ~ 32

Author(s):

Silvia Bartolucci ◽

Michele Mari ◽

Annalida Bedini ◽

Giovanni Piersanti ◽

Gilberto Spadoni

Keyword(s):

Alkylating Agents ◽

Direct Synthesis ◽

Amino Alcohols

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ChemInform Abstract: Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents.

ChemInform ◽

10.1002/chin.201531163 ◽

2015 ◽

Vol 46 (31) ◽

pp. no-no

Author(s):

Silvia Bartolucci ◽

Michele Mari ◽

Annalida Bedini ◽

Giovanni Piersanti ◽

Gilberto Spadoni

Keyword(s):

Alkylating Agents ◽

Direct Synthesis ◽

Amino Alcohols

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ChemInform Abstract: Direct Synthesis of Pyridines and Quinolines by Coupling of γ-Amino-alcohols with Secondary Alcohols Liberating H2Catalyzed by Ruthenium Pincer Complexes.

ChemInform ◽

10.1002/chin.201344154 ◽

2013 ◽

Vol 44 (44) ◽

pp. no-no

Author(s):

Dipankar Srimani ◽

Yehoshoa Ben-David ◽

David Milstein

Keyword(s):

Direct Synthesis ◽

Amino Alcohols ◽

Pincer Complexes ◽

Secondary Alcohols

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The Efficient Direct Synthesis of N,O-Acetal Compounds as Key Intermediates of Discorhabdin A: Oxidative Fragmentation Reaction of α-Amino Acids or β-Amino Alcohols by Using Hypervalent Iodine(III) Reagents.

ChemInform ◽

10.1002/chin.200643025 ◽

2006 ◽

Vol 37 (43) ◽

Author(s):

Yu Harayama ◽

Masako Yoshida ◽

Daigo Kamimura ◽

Yasufumi Wada ◽

Yasuyuki Kita

Keyword(s):

Amino Acids ◽

Direct Synthesis ◽

Amino Alcohols ◽

Hypervalent Iodine ◽

Fragmentation Reaction

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Direct synthesis of N-substituted 1,3-oxazolidines via a hetero-domino Petasis borono-Mannich reaction of 1,2-amino alcohols, formaldehyde, and organoboronic acids

Chemistry of Heterocyclic Compounds ◽

10.1007/s10593-019-02511-8 ◽

2019 ◽

Vol 55 (7) ◽

pp. 648-653 ◽

Cited By ~ 2

Author(s):

Yiting Zheng ◽

Lu Sun ◽

Jiayi Wang ◽

Gonghua Song

Keyword(s):

Mannich Reaction ◽

Direct Synthesis ◽

Amino Alcohols ◽

Organoboronic Acids

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Direct synthesis of pyridines and quinolines by coupling of γ-amino-alcohols with secondary alcohols liberating H2 catalyzed by ruthenium pincer complexes

Chemical Communications ◽

10.1039/c3cc43227k ◽

2013 ◽

Vol 49 (59) ◽

pp. 6632 ◽

Cited By ~ 115

Author(s):

Dipankar Srimani ◽

Yehoshoa Ben-David ◽

David Milstein

Keyword(s):

Direct Synthesis ◽

Amino Alcohols ◽

Pincer Complexes ◽

Secondary Alcohols

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The Efficient Direct Synthesis of N,O-Acetal Compounds as Key Intermediates of Discorhabdin A: Oxidative Fragmentation Reaction of α-Amino Acids or β-Amino Alcohols by Using Hypervalent Iodine(III) Reagents

Chemistry - A European Journal ◽

10.1002/chem.200501635 ◽

2006 ◽

Vol 12 (18) ◽

pp. 4893-4899 ◽

Cited By ~ 27

Author(s):

Yu Harayama ◽

Masako Yoshida ◽

Daigo Kamimura ◽

Yasufumi Wada ◽

Yasuyuki Kita

Keyword(s):

Amino Acids ◽

Direct Synthesis ◽

Amino Alcohols ◽

Hypervalent Iodine ◽

Fragmentation Reaction

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Direct Synthesis of Cyanopyrrolidinyl β-Amino Alcohols for the Development of Diabetes Therapeutics

European Journal of Organic Chemistry ◽

10.1002/ejoc.201600969 ◽

2016 ◽

Vol 2016 (30) ◽

pp. 5160-5168 ◽

Cited By ~ 3

Author(s):

Joseph R. Lizza ◽

Savan V. Patel ◽

Catherine F. Yang ◽

Gustavo Moura-Letts

Keyword(s):

Direct Synthesis ◽

Amino Alcohols

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Multiple myeloma and acute leukemia associated with alkylating agents

Archives of Internal Medicine ◽

10.1001/archinte.135.1.185 ◽

1975 ◽

Vol 135 (1) ◽

pp. 185-192 ◽

Cited By ~ 12

Author(s):

R. A. Kyle

Keyword(s):

Multiple Myeloma ◽

Acute Leukemia ◽

Alkylating Agents

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Diastereoselective synthesis of β-amino alcohols with two or three chiral centers.

Tetrahedron Letters ◽

10.1016/s0040-4039(01)94542-3 ◽

1979 ◽

Vol 19 (15) ◽

pp. 1355-1356

Author(s):

R Haro-Ramos

Keyword(s):

Amino Alcohols ◽

Diastereoselective Synthesis ◽

Chiral Centers

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Standard enthalpies of formation of some refractory borides of 4d and 5d elements from high-temperature direct synthesis calorimetry

Journal de Chimie Physique ◽

10.1051/jcp/1993900349 ◽

1993 ◽

Vol 90 ◽

pp. 349-354 ◽

Cited By ~ 27

Author(s):

SV Meschel ◽

OJ Kleppa

Keyword(s):

High Temperature ◽

Direct Synthesis ◽

Enthalpies Of Formation ◽

Standard Enthalpies Of Formation

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