Structure-based drug screening for G-protein-coupled receptors

Brian K. Shoichet; Brian K. Kobilka

doi:10.1016/j.tips.2012.03.007

Structure-based drug screening for G-protein-coupled receptors

Trends in Pharmacological Sciences ◽

10.1016/j.tips.2012.03.007 ◽

2012 ◽

Vol 33 (5) ◽

pp. 268-272 ◽

Cited By ~ 199

Author(s):

Brian K. Shoichet ◽

Brian K. Kobilka

Keyword(s):

G Protein ◽

Drug Screening ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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A Novel Drug Screening Assay for G Protein‐coupled Receptors

Ligand Design for G Protein‐coupled Receptors - Methods and Principles in Medicinal Chemistry ◽

10.1002/3527608249.ch3 ◽

2006 ◽

pp. 51-60 ◽

Cited By ~ 1

Author(s):

Brian F. O'Dowd ◽

Xiaodong Ji ◽

Mohammad Alijaniaram ◽

Tuan Nguyen ◽

Susan R. George

Keyword(s):

G Protein ◽

Drug Screening ◽

G Protein Coupled Receptors ◽

Screening Assay ◽

Drug Screening Assay ◽

Novel Drug ◽

G Protein Coupled

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Bioluminescence in G Protein-Coupled Receptors Drug Screening Using Nanoluciferase and Halo-Tag Technology

Methods in Molecular Biology - G Protein-Coupled Receptor Screening Assays ◽

10.1007/978-1-0716-1221-7_9 ◽

2021 ◽

pp. 137-147

Author(s):

Hannes Schihada ◽

Katarina Nemec ◽

Martin J. Lohse ◽

Isabella Maiellaro

Keyword(s):

G Protein ◽

Drug Screening ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Selection of In Silico Drug Screening Results for G-Protein-Coupled Receptors by Using Universal Active Probes

Journal of Chemical Information and Modeling ◽

10.1021/ci200236x ◽

2011 ◽

Vol 51 (9) ◽

pp. 2398-2407 ◽

Cited By ~ 17

Author(s):

Mitsuhito Wada ◽

Eiji Kanamori ◽

Haruki Nakamura ◽

Yoshifumi Fukunishi

Keyword(s):

G Protein ◽

Drug Screening ◽

In Silico ◽

G Protein Coupled Receptors ◽

G Protein Coupled ◽

Selection Of

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Oligomerization in Health and Disease: From Enzymes to G Protein-Coupled Receptors

10.1016/s1877-1173(20)x0002-0 ◽

2020 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

Health And Disease ◽

G Protein Coupled

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G Protein-Coupled Receptors Part A

10.1016/s0091-679x(17)x0006-x ◽

2017 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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G Protein-Coupled Receptors - Signaling, Trafficking and Regulation

10.1016/s0091-679x(16)x0002-7 ◽

2016 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Enhanced Salmonella virulence instigated by bactivorous protozoa and investigation of putative protozoan G protein-coupled receptors associated with bacterial engulfment

10.31274/etd-180810-61 ◽

2014 ◽

Author(s):

Matt T. Brewer

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

Salmonella Virulence ◽

G Protein Coupled

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Faculty Opinions recommendation of Modulation of postendocytic sorting of G protein-coupled receptors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1008239.104108 ◽

2002 ◽

Author(s):

Silvia Arber

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Faculty Opinions recommendation of Proteochemometrics modeling of the interaction of amine G-protein coupled receptors with a diverse set of ligands.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1007831.98556 ◽

2002 ◽

Author(s):

Wolfgang Guba

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Faculty Opinions recommendation of Measurement of the millisecond activation switch of G protein-coupled receptors in living cells.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1014169.192885 ◽

2003 ◽

Author(s):

Kees Jalink

Keyword(s):

G Protein ◽

Living Cells ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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