Dimerization of β-tryptase inhibitors, does it work for both basic and neutral P1 groups?

2012 ◽  
Vol 22 (9) ◽  
pp. 3370-3376 ◽  
Author(s):  
Guyan Liang ◽  
Yong Mi Choi-Sledeski ◽  
Xin Chen ◽  
Yong Gong ◽  
Eric W. MacMillan ◽  
...  
Keyword(s):  
Tryptase Inhibitors

Synthesis and evaluation of 4-substituted benzylamine derivatives as β-tryptase inhibitors

2006 ◽  
Vol 16 (11) ◽  
pp. 2986-2990 ◽  
Author(s):  
Yutaka Miyazaki ◽  
Yutaka Kato ◽  
Tadashi Manabe ◽  
Hiroyasu Shimada ◽  
Masashi Mizuno ◽  
...  
Keyword(s):  
Tryptase Inhibitors

Tryptase inhibitors: a novel class of anti-inflammatory drugs

1997 ◽  
Vol 6 (7) ◽  
pp. 811-817 ◽  
Author(s):  
Robert P Numerof ◽  
Paul J Simpson ◽  
Richard Tanaka
Keyword(s):  
Inflammatory Drugs ◽  
Anti Inflammatory ◽  
Tryptase Inhibitors

Design, synthesis and biological activity of a targeted library of potential tryptase inhibitors

2004 ◽  
Vol 2 (11) ◽  
pp. 1633-1642 ◽  
Author(s):  
Mónica García ◽  
Xavier del Río ◽  
Sandra Silvestre ◽  
Mario Rubiralta ◽  
Estrella Lozoya ◽  
...  
Keyword(s):  
Biological Activity ◽  
Design Synthesis ◽  
Tryptase Inhibitors ◽  
Targeted Library

Synthesis and SAR of 4-Carboxy-2-azetidinone Mechanism-Based Tryptase Inhibitors (I).

ChemInform ◽  
2003 ◽  
Vol 34 (8) ◽  
Author(s):  
James C. Sutton ◽  
et al. et al.
Keyword(s):  
Tryptase Inhibitors

Design and Synthesis of Selective Keto-1,2,4-oxadiazole-based Tryptase Inhibitors.

ChemInform ◽  
2006 ◽  
Vol 37 (38) ◽  
Author(s):  
James T. Palmer ◽  
Robert M. Rydzewski ◽  
Rohan V. Mendonca ◽  
David Sperandio ◽  
Jeffrey R. Spencer ◽  
...  
Keyword(s):  
Design And Synthesis ◽  
Tryptase Inhibitors

Tryptase inhibitors block allergen-induced airway and inflammatory responses in allergic sheep.

1995 ◽  
Vol 152 (6) ◽  
pp. 2076-2083 ◽  
Author(s):  
J M Clark ◽  
W M Abraham ◽  
C E Fishman ◽  
R Forteza ◽  
A Ahmed ◽  
...  
Keyword(s):  
Inflammatory Responses ◽  
Tryptase Inhibitors

Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors

2006 ◽  
Vol 16 (13) ◽  
pp. 3434-3439 ◽  
Author(s):  
James T. Palmer ◽  
Robert M. Rydzewski ◽  
Rohan V. Mendonca ◽  
David Sperandio ◽  
Jeffrey R. Spencer ◽  
...  
Keyword(s):  
Design And Synthesis ◽  
Tryptase Inhibitors

Cyclotheonamide E4 and E5, New Potent Tryptase Inhibitors from anIrciniaSpecies of Sponge

2002 ◽  
Vol 65 (3) ◽  
pp. 259-261 ◽  
Author(s):  
Yasunobu Murakami ◽  
Masao Takei ◽  
Kazutoshi Shindo ◽  
Chie Kitazume ◽  
Junichi Tanaka ◽  
...  
Keyword(s):  
Tryptase Inhibitors
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