Synthesis and structure–activity relationships of 4,5-fused pyridazinones as histamine H3 receptor antagonists

2011 ◽  
Vol 21 (20) ◽  
pp. 6126-6130 ◽  
Author(s):  
Ming Tao ◽  
Rita Raddatz ◽  
Lisa D. Aimone ◽  
Robert L. Hudkins
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists.

ChemInform ◽  
2000 ◽  
Vol 31 (40) ◽  
pp. no-no
Author(s):  
Ian D. Linney ◽  
Ildiko M. Buck ◽  
Elaine A. Harper ◽  
S. Barret-Kalindjian ◽  
Michael J. Pether ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Novel Histamine H3-Receptor Antagonists with Benzyl Ether Structure or Related Moieties: Synthesis and Structure-Activity Relationships

1996 ◽  
Vol 329 (8-9) ◽  
pp. 379-385 ◽  
Author(s):  
Annette Hüls ◽  
Katja Purand ◽  
Holger Stark ◽  
Sibylle Reidemeister ◽  
Xavier Ligneau ◽  
...  
Keyword(s):  
Benzyl Ether ◽  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists

2005 ◽  
Vol 13 (19) ◽  
pp. 5647-5657 ◽  
Author(s):  
Simone Lorenzi ◽  
Marco Mor ◽  
Fabrizio Bordi ◽  
Silvia Rivara ◽  
Mirko Rivara ◽  
...  
Keyword(s):  
Receptor Model ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Synthesis, structure–activity relationships, and biological profiles of a dihydrobenzoxathiin class of histamine H3 receptor inverse agonists

2009 ◽  
Vol 19 (15) ◽  
pp. 4232-4236 ◽  
Author(s):  
Takahide Sasaki ◽  
Toshiyuki Takahashi ◽  
Tsuyoshi Nagase ◽  
Takashi Mizutani ◽  
Sayaka Ito ◽  
...  
Keyword(s):  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Synthesis and structure–activity relationships of N-aryl-piperidine derivatives as potent (partial) agonists for human histamine H3 receptor

2010 ◽  
Vol 18 (14) ◽  
pp. 5441-5448 ◽  
Author(s):  
Makoto Ishikawa ◽  
Takeshi Furuuchi ◽  
Miki Yamauchi ◽  
Fumikazu Yokoyama ◽  
Nobukazu Kakui ◽  
...  
Keyword(s):  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Partial Agonists ◽  
Structure Activity ◽  
H3 Receptor ◽  
Human Histamine ◽  
Histamine H3
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