Azepanone-based inhibitors of human cathepsin S: Optimization of selectivity via the P2 substituent

2011 ◽  
Vol 21 (15) ◽  
pp. 4409-4415 ◽  
Author(s):  
Jeffrey K. Kerns ◽  
Hong Nie ◽  
William Bondinell ◽  
Katherine L. Widdowson ◽  
Dennis S. Yamashita ◽  
...  
Keyword(s):  
Cathepsin S ◽  
Human Cathepsin

scholarly journals Crystal structure of human cathepsin S

1998 ◽  
Vol 7 (6) ◽  
pp. 1294-1302 ◽  
Author(s):  
Mary E. Mcgrath ◽  
James T. Palmer ◽  
Ddeter Brömme ◽  
John R. Somoza
Keyword(s):  
Crystal Structure ◽  
Cathepsin S ◽  
Human Cathepsin

scholarly journals High level expression and crystallization of recombinant human cathepsin S

1996 ◽  
Vol 5 (4) ◽  
pp. 789-791 ◽  
Author(s):  
Dieter Brömme ◽  
Mary E. Mcgrath
Keyword(s):  
Cathepsin S ◽  
High Level Expression ◽  
Human Cathepsin ◽  
High Level

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

2018 ◽  
Vol 26 (14) ◽  
pp. 4310-4319 ◽  
Author(s):  
Zahira Tber ◽  
Mylène Wartenberg ◽  
Jean-Eddy Jacques ◽  
Vincent Roy ◽  
Fabien Lecaille ◽  
...  
Keyword(s):  
Selective Inhibition ◽  
Cathepsin S ◽  
Human Cathepsin

Structure of a Cys25→Ser mutant of human cathepsin S

2002 ◽  
Vol 58 (3) ◽  
pp. 451-455 ◽  
Author(s):  
Johan P. Turkenburg ◽  
Marieke B. A. C. Lamers ◽  
A. Marek Brzozowski ◽  
Lisa M. Wright ◽  
Roderick E. Hubbard ◽  
...  
Keyword(s):  
Cathepsin S ◽  
Human Cathepsin

Controlled Peptide Solvation in Portion-Mixing Libraries of FRET Peptides:  Improved Specificity Determination for Dengue 2 Virus NS2B-NS3 Protease and Human Cathepsin S

2007 ◽  
Vol 9 (4) ◽  
pp. 627-634 ◽  
Author(s):  
Fabiana M. Alves ◽  
Izaura Y. Hirata ◽  
Iuri E. Gouvea ◽  
Marcio F. M. Alves ◽  
Morten Meldal ◽  
...  
Keyword(s):  
Cathepsin S ◽  
Human Cathepsin ◽  
Ns3 Protease

scholarly journals Phylogenetic conservation of cysteine proteinases. Cloning and expression of a cDNA coding for human cathepsin S.

1992 ◽  
Vol 267 (19) ◽  
pp. 13708-13713 ◽  
Author(s):  
B Wiederanders ◽  
D Brömme ◽  
H Kirschke ◽  
K von Figura ◽  
B Schmidt ◽  
...  
Keyword(s):  
Cloning And Expression ◽  
Cathepsin S ◽  
Cysteine Proteinases ◽  
Phylogenetic Conservation ◽  
Human Cathepsin

scholarly journals Human cathepsin S gene (CTSS) promoter −25G/A polymorphism

2000 ◽  
Vol 45 (2) ◽  
pp. 94-95 ◽  
Author(s):  
Henian Cao ◽  
Robert A. Hegele
Keyword(s):  
Cathepsin S ◽  
S Gene ◽  
Human Cathepsin

N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S: In silico design, synthesis and biochemical characterization

2020 ◽  
Vol 30 (18) ◽  
pp. 127420
Author(s):  
Carina Lemke ◽  
Lorenzo Cianni ◽  
Christian Feldmann ◽  
Erik Gilberg ◽  
Jiafei Yin ◽  
...  
Keyword(s):  
In Silico ◽  
Biochemical Characterization ◽  
Cathepsin S ◽  
Design Synthesis ◽  
In Silico Design ◽  
Human Cathepsin
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