Synthesis and receptor binding properties of chimeric peptides containing a μ-opioid receptor ligand and nociceptin/orphanin FQ receptor ligand Ac-RYYRIK-amide

Susumu Kawano; Akihiro Ambo; Yusuke Sasaki

doi:10.1016/j.bmcl.2006.06.060

Synthesis and receptor binding properties of chimeric peptides containing a μ-opioid receptor ligand and nociceptin/orphanin FQ receptor ligand Ac-RYYRIK-amide

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.06.060 ◽

2006 ◽

Vol 16 (18) ◽

pp. 4839-4841 ◽

Cited By ~ 9

Author(s):

Susumu Kawano ◽

Akihiro Ambo ◽

Yusuke Sasaki

Keyword(s):

Opioid Receptor ◽

Receptor Binding ◽

Orphanin Fq ◽

Binding Properties ◽

Receptor Ligand ◽

Μ Opioid Receptor ◽

Chimeric Peptides

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Receptor Binding Properties and Antinociceptive Effects of Chimeric Peptides Consisting of a μ-Opioid Receptor Agonist and an ORL1 Receptor Antagonist

Biological and Pharmaceutical Bulletin ◽

10.1248/bpb.30.1260 ◽

2007 ◽

Vol 30 (7) ◽

pp. 1260-1264 ◽

Cited By ~ 9

Author(s):

Susumu Kawano ◽

Risa Ito ◽

Miharu Nishiyama ◽

Mai Kubo ◽

Tomoko Matsushima ◽

...

Keyword(s):

Receptor Antagonist ◽

Opioid Receptor ◽

Receptor Binding ◽

Receptor Agonist ◽

Mu Opioid Receptor ◽

Binding Properties ◽

Mu Opioid ◽

Opioid Receptor Agonist ◽

Antinociceptive Effects ◽

Chimeric Peptides

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Redefining the structure–activity relationships of 2,6-methano-3-benzazocines. Part 6: Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocine

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.03.066 ◽

2008 ◽

Vol 16 (10) ◽

pp. 5653-5664 ◽

Cited By ~ 5

Author(s):

Mark P. Wentland ◽

Xufeng Sun ◽

Dana J. Cohen ◽

Jean M. Bidlack

Keyword(s):

Opioid Receptor ◽

Receptor Binding ◽

Binding Properties ◽

Structure Activity Relationships ◽

Structure Activity ◽

Opioid Receptor Binding Properties ◽

Opioid Receptor Binding

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Chronic ethanol alters the receptor binding characteristics of the delta opioid receptor ligand, DAla2DLeu5 enkephalin in mouse brain

Life Sciences ◽

10.1016/0024-3205(83)90267-9 ◽

1983 ◽

Vol 33 (23) ◽

pp. 2331-2337 ◽

Cited By ~ 42

Author(s):

Martin D. Hynes ◽

Mary Ann Lochner ◽

Kerry G. Bemis ◽

David L. Hymson

Keyword(s):

Opioid Receptor ◽

Mouse Brain ◽

Receptor Binding ◽

Chronic Ethanol ◽

Delta Opioid Receptor ◽

Receptor Ligand ◽

Binding Characteristics

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Redefining the structure–activity relationships of 2,6-methano-3-benzazocines. 5. Opioid receptor binding properties of N-((4′-phenyl)-phenethyl) analogues of 8-CAC

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.09.082 ◽

2007 ◽

Vol 17 (23) ◽

pp. 6516-6520 ◽

Cited By ~ 9

Author(s):

Melissa A. VanAlstine ◽

Mark P. Wentland ◽

Dana J. Cohen ◽

Jean M. Bidlack

Keyword(s):

Opioid Receptor ◽

Receptor Binding ◽

Binding Properties ◽

Structure Activity Relationships ◽

Structure Activity ◽

Opioid Receptor Binding Properties ◽

Opioid Receptor Binding

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Opioid receptor binding properties of [3H]Buprenorphine in rat brain

European Neuropsychopharmacology ◽

10.1016/0924-977x(96)87980-6 ◽

1996 ◽

Vol 6 ◽

pp. 146-147

Author(s):

A. Borsodi ◽

F. Ötvös ◽

G. Tóth ◽

S. Hosztafi ◽

C. Simon ◽

...

Keyword(s):

Rat Brain ◽

Opioid Receptor ◽

Receptor Binding ◽

Binding Properties ◽

Opioid Receptor Binding Properties ◽

Opioid Receptor Binding

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Painful Inflammation-Induced Increase in μ-Opioid Receptor Binding and G-Protein Coupling in Primary Afferent Neurons

Molecular Pharmacology ◽

10.1124/mol.64.2.202 ◽

2003 ◽

Vol 64 (2) ◽

pp. 202-210 ◽

Cited By ~ 136

Author(s):

C. Zöllner ◽

M. A. Shaqura ◽

C. P. Bopaiah ◽

S. Mousa ◽

C. Stein ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Receptor Binding ◽

Afferent Neurons ◽

G Protein Coupling ◽

Primary Afferent Neurons ◽

Primary Afferent ◽

Protein Coupling ◽

Μ Opioid Receptor ◽

Opioid Receptor Binding

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Structural Basis for μ-Opioid Receptor Binding and Activation

Structure ◽

10.1016/j.str.2011.08.003 ◽

2011 ◽

Vol 19 (11) ◽

pp. 1683-1690 ◽

Cited By ~ 17

Author(s):

Adrian W.R. Serohijos ◽

Shuangye Yin ◽

Feng Ding ◽

Josee Gauthier ◽

Dustin G. Gibson ◽

...

Keyword(s):

Opioid Receptor ◽

Receptor Binding ◽

Structural Basis ◽

Μ Opioid Receptor ◽

Opioid Receptor Binding

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GABAA and μ-opioid receptor binding in the globus pallidus and entopeduncular nucleus of animals symptomatic for and recovered from experimental Parkinsonism

Brain Research ◽

10.1016/s0006-8993(02)03010-x ◽

2002 ◽

Vol 947 (2) ◽

pp. 284-289 ◽

Cited By ~ 5

Author(s):

Joseph A Schroeder ◽

Jay S Schneider

Keyword(s):

Globus Pallidus ◽

Opioid Receptor ◽

Receptor Binding ◽

Entopeduncular Nucleus ◽

Experimental Parkinsonism ◽

Μ Opioid Receptor ◽

Opioid Receptor Binding

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Redefining the Structure−Activity Relationships of 2,6-Methano-3-benzazocines. 4. Opioid Receptor Binding Properties of 8-[N-(4‘-phenyl)-phenethyl)carboxamido] Analogues of Cyclazocine and Ethylketocycalzocine

Journal of Medicinal Chemistry ◽

10.1021/jm060278n ◽

2006 ◽

Vol 49 (18) ◽

pp. 5635-5639 ◽

Cited By ~ 19

Author(s):

Mark P. Wentland ◽

Melissa VanAlstine ◽

Robert Kucejko ◽

Rongliang Lou ◽

Dana J. Cohen ◽

...

Keyword(s):

Opioid Receptor ◽

Receptor Binding ◽

Binding Properties ◽

Structure Activity Relationships ◽

Structure Activity ◽

Opioid Receptor Binding Properties ◽

Opioid Receptor Binding

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Molecular modeling of salsolinol, a full G i protein agonist of the μ‐opioid receptor, within the receptor binding site

Chemical Biology & Drug Design ◽

10.1111/cbdd.13523 ◽

2019 ◽

Cited By ~ 1

Author(s):

Pablo Berríos‐Cárcamo ◽

Mario Rivera‐Meza ◽

Mario Herrera‐Marschitz ◽

Gerald Zapata‐Torres

Keyword(s):

Molecular Modeling ◽

Binding Site ◽

Opioid Receptor ◽

Receptor Binding ◽

Receptor Binding Site ◽

Μ Opioid Receptor

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