Synthesis and pharmacological studies of new hybrid derivatives of fentanyl active at the μ-opioid receptor and I2–imidazoline binding sites

2006 ◽  
Vol 14 (19) ◽  
pp. 6570-6580 ◽  
Author(s):  
Christophe Dardonville ◽  
Cristina Fernandez-Fernandez ◽  
Sarah-Louise Gibbons ◽  
Gary J. Ryan ◽  
Nadine Jagerovic ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Binding Sites ◽  
Pharmacological Studies ◽  
Μ Opioid Receptor ◽  
Imidazoline Binding Sites ◽  
Derivatives Of

Refinement of a Homology Model of the μ-Opioid Receptor Using Distance Constraints from Intrinsic and Engineered Zinc-Binding Sites†

Biochemistry ◽  
2004 ◽  
Vol 43 (27) ◽  
pp. 8700-8710 ◽  
Author(s):  
Carol B. Fowler ◽  
Irina D. Pogozheva ◽  
Harry LeVine ◽  
Henry I. Mosberg
Keyword(s):  
Opioid Receptor ◽  
Binding Sites ◽  
Homology Model ◽  
Zinc Binding ◽  
Distance Constraints ◽  
Μ Opioid Receptor

Identification of Endomorphin-1 and Endomorphin-2 Binding Sites in Human μ-Opioid Receptor by Antisense Oligonucleotide Strategy

2008 ◽  
Vol 72 (6) ◽  
pp. 507-512 ◽  
Author(s):  
Jakub Fichna ◽  
Katarzyna Gach ◽  
Renata Perlikowska ◽  
Jeroen Poels ◽  
Jozef Vanden Broeck ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Binding Sites ◽  
Antisense Oligonucleotide ◽  
Μ Opioid Receptor

μ-Opioid receptor and α2-adrenoceptor agonist binding sites in the postmortem brain of heroin addicts

1994 ◽  
Vol 115 (1-2) ◽  
pp. 135-140 ◽  
Author(s):  
Ane M. Gabilondo ◽  
J. Javier Meana ◽  
Fernando Barturen ◽  
Magdalena Sastre ◽  
Jesús A. García-Sevilla
Keyword(s):  
Opioid Receptor ◽  
Binding Sites ◽  
Postmortem Brain ◽  
Agonist Binding ◽  
Heroin Addicts ◽  
Α2 Adrenoceptor ◽  
Adrenoceptor Agonist ◽  
Μ Opioid Receptor

Ligand recognition in μ opioid receptor: experimentally based modeling of μ opioid receptor binding sites and their testing by ligand docking

1996 ◽  
Vol 4 (12) ◽  
pp. 2151-2166 ◽  
Author(s):  
Takeshi Sagara ◽  
Hiromu Egashira ◽  
Mikako Okamura ◽  
Ikuo Fujii ◽  
Yasuyuki Shimohigashi ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Receptor Binding ◽  
Binding Sites ◽  
Ligand Docking ◽  
Ligand Recognition ◽  
Μ Opioid Receptor ◽  
Opioid Receptor Binding

14β-Chlorocinnamoylamino derivatives of metopon: long-term μ-opioid receptor antagonists

1997 ◽  
Vol 320 (2-3) ◽  
pp. 121-129 ◽  
Author(s):  
Jay P McLaughlin ◽  
Alice Sebastian ◽  
Sydney Archer ◽  
Jean M Bidlack
Keyword(s):  
Opioid Receptor ◽  
Receptor Antagonists ◽  
Opioid Receptor Antagonists ◽  
Μ Opioid Receptor ◽  
Derivatives Of
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