Antimuscarinic, calcium channel blocker and tachykinin NK2 receptor antagonist actions of otilonium bromide in the circular muscle of guinea-pig colon

1999 ◽  
Vol 359 (5) ◽  
pp. 420-427 ◽  
Author(s):  
P. Santicioli ◽  
Vladimir Zagorodnyuk ◽  
Anna Rita Renzetti ◽  
Carlo Alberto Maggi
Keyword(s):  
Guinea Pig ◽  
Calcium Channel ◽  
Receptor Antagonist ◽  
Calcium Channel Blocker ◽  
Channel Blocker ◽  
Circular Muscle ◽  
Nk2 Receptor ◽  
Tachykinin Nk2 Receptor

MEN 11420, a potent and selective tachykinin NK2 receptor antagonist in the guinea-pig and human colon

1997 ◽  
Vol 356 (5) ◽  
pp. 678-688 ◽  
Author(s):  
Paolo Santicioli ◽  
Sandro Giuliani ◽  
Riccardo Patacchini ◽  
Manuela Tramontana ◽  
Marco Criscuoli ◽  
...  
Keyword(s):  
Guinea Pig ◽  
Receptor Antagonist ◽  
Human Colon ◽  
Nk2 Receptor ◽  
Tachykinin Nk2 Receptor

scholarly journals Angiotensin-II receptor antagonist combined with calcium channel blocker or diuretic for essential hypertension

2009 ◽  
Vol 32 (11) ◽  
pp. 962-968 ◽  
Author(s):  
Toshihiko Ishimitsu ◽  
Atsushi Numabe ◽  
Toshihide Masuda ◽  
Tomoyuki Akabane ◽  
Atsushi Okamura ◽  
...  
Keyword(s):  
Essential Hypertension ◽  
Angiotensin Ii ◽  
Calcium Channel ◽  
Receptor Antagonist ◽  
Calcium Channel Blocker ◽  
Channel Blocker ◽  
Angiotensin Ii Receptor ◽  
Angiotensin Ii Receptor Antagonist

Antibronchospastic activity of MEN10,627, a novel tachykinin NK2 receptor antagonist, in guinea-pig airways

1995 ◽  
Vol 273 (1-2) ◽  
pp. 129-135 ◽  
Author(s):  
Francesca Perretti ◽  
Lido Ballati ◽  
Stefano Manzini ◽  
Carlo Alberto Maggi ◽  
Stefano Evangelista
Keyword(s):  
Guinea Pig ◽  
Receptor Antagonist ◽  
Nk2 Receptor ◽  
Tachykinin Nk2 Receptor

Radiosynthesis of dimethyl-2-[18F]-(fluoromethyl)-6-methyl-4-(2-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate for L-type calcium channel imaging

2008 ◽  
Vol 96 (12) ◽  
Author(s):  
H. Sadeghpour ◽  
A. R. Jalilian ◽  
A. Shafiee ◽  
M. Akhlaghi ◽  
R. Miri ◽  
...  
Keyword(s):  
Smooth Muscle ◽  
Guinea Pig ◽  
Calcium Channel ◽  
Calcium Channel Blocker ◽  
Channel Blocker ◽  
Muscle Model ◽  
Channel Distribution ◽  
Longitudinal Smooth Muscle ◽  
Biological Studies

AbstractDimethyl 2-(fluoromethyl)-6-methyl-4-(2-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate 4a, a fluorinated nifedipine analog, has been shown to elicit significant calcium channel blocker activity using a guinea pig ileal longitudinal smooth muscle model. In order to perform biological studies for detection of L-type calcium channel distribution, we decided to prepare the [

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