Medicinal Chemistry of σ1 Receptor Ligands: Pharmacophore Models, Synthesis, Structure Affinity Relationships, and Pharmacological Applications

2017 ◽  
pp. 51-79 ◽  
Author(s):  
Frauke Weber ◽  
Bernhard Wünsch
Keyword(s):  
Medicinal Chemistry ◽  
Receptor Ligands ◽  
Σ1 Receptor ◽  
Pharmacophore Models

scholarly journals Recent Advances in the Development of Sigma Receptor Ligands as Cytotoxic Agents: A Medicinal Chemistry Perspective

2021 ◽  
Author(s):  
Antonino N. Fallica ◽  
Valeria Pittalà ◽  
Maria N. Modica ◽  
Loredana Salerno ◽  
Giuseppe Romeo ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Cytotoxic Agents ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Sigma Receptor Ligands ◽  
Recent Advances

5D-QSAR for spirocyclic σ1 receptor ligands by Quasar receptor surface modeling

2010 ◽  
Vol 45 (7) ◽  
pp. 3116-3124 ◽  
Author(s):  
Christoph Oberdorf ◽  
Thomas J. Schmidt ◽  
Bernhard Wünsch
Keyword(s):  
Surface Modeling ◽  
Receptor Ligands ◽  
Σ1 Receptor

scholarly journals The Medicinal Chemistry of 5-HT6 Receptor Ligands with a Focus on Arylsulfonyltryptamine Analogs

2010 ◽  
Vol 10 (5) ◽  
pp. 579-595 ◽  
Author(s):  
Richard A. Glennon ◽  
Uma Siripurapu ◽  
Bryan L. Roth ◽  
Renata Kolanos ◽  
Mikhail L. Bondarev ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Receptor Ligands

The Medicinal Chemistry of 5-HT2C Receptor Ligands

2010 ◽  
pp. 29-50
Author(s):  
Marcello Leopoldo ◽  
Enza Lacivita ◽  
Paola De Giorgio ◽  
Francesco Berardi ◽  
Roberto Perrone
Keyword(s):  
Medicinal Chemistry ◽  
Receptor Ligands

Predicting the Antinociceptive Efficacy of σ1 Receptor Ligands by a Novel Receptor Fluorescence Resonance Energy Transfer (FRET) Based Biosensor

2013 ◽  
Vol 57 (1) ◽  
pp. 238-242 ◽  
Author(s):  
Maricel Gómez-Soler ◽  
Víctor Fernández-Dueñas ◽  
Enrique Portillo-Salido ◽  
Pilar Pérez ◽  
Daniel Zamanillo ◽  
...  
Keyword(s):  
Energy Transfer ◽  
Fluorescence Resonance Energy Transfer ◽  
Resonance Energy Transfer ◽  
Resonance Energy ◽  
Receptor Ligands ◽  
Σ1 Receptor ◽  
Fluorescence Resonance

Synthesis and Structure–Activity Relationship Study of a New Series of Selective σ1 Receptor Ligands for the Treatment of Pain: 4-Aminotriazoles

2015 ◽  
Vol 58 (5) ◽  
pp. 2441-2451 ◽  
Author(s):  
José Luis Díaz ◽  
Ute Christmann ◽  
Ariadna Fernández ◽  
Antoni Torrens ◽  
Adriana Port ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Receptor Ligands ◽  
Σ1 Receptor ◽  
Structure Activity ◽  
Relationship Study
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