Water‐Promoted Synthesis of Azepino[3,4,5‐ cd ]indole Analogues via Pictet‐Spengler Reaction

2020 ◽  
Vol 5 (15) ◽  
pp. 4619-4622
Author(s):  
Shuaizhong Zhang ◽  
Yunrui Cai ◽  
Hongbin Zou
Keyword(s):  
Indole Analogues

Synthesis, antimicrobial, and antioxidant activities of some new indole analogues containing pyrimidine and fused pyrimidine systems

2011 ◽  
Vol 21 (11) ◽  
pp. 3809-3817 ◽  
Author(s):  
Saundane Anand Raghunath ◽  
Yarlakatti Manjunatha ◽  
Kalpana Rayappa
Keyword(s):  
Antioxidant Activities ◽  
Indole Analogues

Synthesis and larvicidal properties of benzophenone comprise indole analogues against Culex quinquefasciatus

2013 ◽  
Vol 5 (4) ◽  
pp. 275-280 ◽  
Author(s):  
V. Lakshmi Ranganatha ◽  
A. Bushra Begum ◽  
T. Prashanth ◽  
H.D. Gurupadaswamy ◽  
S.K. Madhu ◽  
...  
Keyword(s):  
Culex Quinquefasciatus ◽  
Indole Analogues

Synthesis of indole analogues of the anti-Helicobacter pylori compounds CJ-13,015, CJ-13,102, CJ-13,104 and CJ-13,108

Tetrahedron ◽  
2007 ◽  
Vol 63 (25) ◽  
pp. 5379-5385 ◽  
Author(s):  
Zoe E. Wilson ◽  
Amanda M. Heapy ◽  
Margaret A. Brimble
Keyword(s):  
Helicobacter Pylori ◽  
Indole Analogues

QSAR Analysis of Indole Analogues as Monoamine Oxidase Inhibitors

1996 ◽  
Vol 36 (4) ◽  
pp. 664-671 ◽  
Author(s):  
A. E. Medvedev ◽  
A. S. Ivanov ◽  
A. V. Veselovsky ◽  
V. S. Skvortsov ◽  
A. I. Archakov
Keyword(s):  
Monoamine Oxidase ◽  
Monoamine Oxidase Inhibitors ◽  
Qsar Analysis ◽  
Indole Analogues

Synthesis and pharmacological evaluation of 1,2,3,4-tetrahydropyrazino[1,2-a]indole and 2-[(phenylmethylamino)methyl]-1H-indole analogues as novel melatoninergic ligands

2009 ◽  
Vol 17 (13) ◽  
pp. 4583-4594 ◽  
Author(s):  
Christian Markl ◽  
Mohamed I. Attia ◽  
Justin Julius ◽  
Shalini Sethi ◽  
Paula A. Witt-Enderby ◽  
...  
Keyword(s):  
Pharmacological Evaluation ◽  
Indole Analogues

scholarly journals Microwave Assisted Synthesis of Novel Imidazolopyridinyl Indoles as Potent Antioxidant and Antimicrobial Agents

2014 ◽  
Vol 2014 ◽  
pp. 1-8 ◽  
Author(s):  
Jaiprakash S. Biradar ◽  
Parveen Rajesab ◽  
Sasidhar B. Somappa
Keyword(s):  
Antimicrobial Agents ◽  
Analytical Data ◽  
Antimicrobial Activities ◽  
Microwave Assisted Synthesis ◽  
The Novel ◽  
Design Synthesis ◽  
Mass Spectral ◽  
H Nmr ◽  
Total Antioxidant ◽  
Indole Analogues

We describe herein the design, synthesis, and pharmacological evaluation of novel series of imidazolopyridinyl indole analogues as potent antioxidants and antimicrobials. These novel compounds (3a–i) were synthesized by reacting 3,5-disubstituted-indole-2-carboxylic acid (1a–i) with 2,3-diamino pyridine (2) in excellent yield. The novel products were confirmed by their IR,1H NMR,13C NMR, mass spectral, and analytical data. These compounds were screened for their antioxidant and antimicrobial activities. Among the compounds tested,3a–dshowed the highest total antioxidant capacity, scavenging, and antimicrobial activities. Compounds3c-dand3g-hhave shown excellent ferric reducing activity.

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