In vivo and in vitro metabolism of the synthetic cannabinoid JWH-200

2013 ◽  
Vol 27 (18) ◽  
pp. 2115-2126 ◽  
Author(s):  
Nik De Brabanter ◽  
Simone Esposito ◽  
Eva Tudela ◽  
Leen Lootens ◽  
Philip Meuleman ◽  
...  
Keyword(s):  
Synthetic Cannabinoid ◽  
In Vitro Metabolism

In vivo and in vitro metabolism of the novel synthetic cannabinoid 5F-APINAC

2019 ◽  
Vol 38 (1) ◽  
pp. 160-171 ◽  
Author(s):  
Svetlana A. Appolonova ◽  
Covadonga Palacio ◽  
Ksenia M. Shestakova ◽  
Natalia V. Mesonzhnik ◽  
Alex Brito ◽  
...  
Keyword(s):  
Synthetic Cannabinoid ◽  
In Vitro Metabolism ◽  
The Novel

scholarly journals GPR18, GPR55 and GPR119 (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

2019 ◽  
Vol 2019 (4) ◽  
Author(s):  
Stephen P.H. Alexander ◽  
Andrew J. Irving
Keyword(s):  
Cannabinoid Receptors ◽  
Cannabinoid Receptor ◽  
Structural Similarity ◽  
Synthetic Cannabinoid ◽  
Receptor Ligands ◽  
Orphan Status ◽  
Endogenous Cannabinoid

GPR18, GPR55 and GPR119 (provisional nomenclature), although showing little structural similarity to CB1 and CB2 cannabinoid receptors, respond to endogenous agents analogous to the endogenous cannabinoid ligands, as well as some natural/synthetic cannabinoid receptor ligands [98]. Although there are multiple reports to indicate that GPR18, GPR55 and GPR119 can be activated in vitro by N-arachidonoylglycine, lysophosphatidylinositol and N-oleoylethanolamide, respectively, there is a lack of evidence for activation by these lipid messengers in vivo. As such, therefore, these receptors retain their orphan status.

Enantioselective in vitro metabolism and in vitro-in vivo correlation of the herbicide ethofumesate in a human model

2020 ◽  
Vol 187 ◽  
pp. 113349 ◽  
Author(s):  
Icaro Salgado Perovani ◽  
Daniel Blascke Carrão ◽  
Nayara Cristina Perez de Albuquerque ◽  
Anderson Rodrigo Moraes de Oliveira
Keyword(s):  
In Vitro Metabolism ◽  
Human Model

In vivo and in vitro metabolism of ethylenethiourea in the rat and the cat

1980 ◽  
Vol 52 (1) ◽  
pp. 16-21 ◽  
Author(s):  
F. Iverson ◽  
K.S. Khera ◽  
S.L. Hierlihy
Keyword(s):  
In Vitro Metabolism
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