Irreversible enzyme inhibitors. XCIV. inhibition of dihydrofolic reductase with derivatives of 2,6-diaminopurines

B. R. Baker; Daniel V. Santi

doi:10.1002/jhet.5570040209

Irreversible enzyme inhibitors. XCIV. inhibition of dihydrofolic reductase with derivatives of 2,6-diaminopurines

Journal of Heterocyclic Chemistry ◽

10.1002/jhet.5570040209 ◽

1967 ◽

Vol 4 (2) ◽

pp. 216-223 ◽

Cited By ~ 4

Author(s):

B. R. Baker ◽

Daniel V. Santi

Keyword(s):

Enzyme Inhibitors ◽

Derivatives Of

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5476847 Derivatives of phosphinic acid useful as endothelin converting enzyme inhibitors

Biotechnology Advances ◽

10.1016/s0734-9750(97)88331-0 ◽

1997 ◽

Vol 15 (1) ◽

pp. 204

Keyword(s):

Enzyme Inhibitors ◽

Phosphinic Acid ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Endothelin Converting Enzyme ◽

Derivatives Of

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Molecular and crystal structures of MDL27,467A hydrochloride and quinapril hydrochloride, two ester derivatives of potent angiotensin converting enzyme inhibitors

Journal of Medicinal Chemistry ◽

10.1021/jm00106a005 ◽

1991 ◽

Vol 34 (2) ◽

pp. 511-517 ◽

Cited By ~ 10

Author(s):

Roland J. Hausin ◽

Penelope W. Codding

Keyword(s):

Angiotensin Converting Enzyme ◽

Crystal Structures ◽

Enzyme Inhibitors ◽

Angiotensin Converting Enzyme Inhibitors ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Molecular And Crystal Structures ◽

Derivatives Of ◽

Quinapril Hydrochloride

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Design, Synthesis, and Evaluation of Acyclic C-Nucleoside and N-Methylated Derivatives of the Ribitylaminopyrimidine Substrate of Lumazine Synthase as Potential Enzyme Inhibitors and Mechanistic Probes.

ChemInform ◽

10.1002/chin.200508222 ◽

2005 ◽

Vol 36 (8) ◽

Author(s):

Jinhua Chen ◽

Thota Sambaiah ◽

Boris Illarionov ◽

Markus Fischer ◽

Adelbert Bacher ◽

...

Keyword(s):

Enzyme Inhibitors ◽

Design Synthesis ◽

Lumazine Synthase ◽

Derivatives Of

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Irreversible enzyme inhibitors. 181. Inhibition of brain choline acetyltransferase by derivatives of 4-stilbazole

Journal of Medicinal Chemistry ◽

10.1021/jm00286a011 ◽

1971 ◽

Vol 14 (4) ◽

pp. 315-322 ◽

Cited By ~ 37

Author(s):

Bernard Randall Baker ◽

Raymond E. Gibson

Keyword(s):

Choline Acetyltransferase ◽

Enzyme Inhibitors ◽

Derivatives Of

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The asymmetric synthesis of arginine mimetics: derivatives of (S)-2-, 3- and 4-amidinophenylalanine suitable for incorporation into enzyme inhibitors and/or peptides

Journal of Peptide Research ◽

10.1111/j.1399-3011.1998.tb01477.x ◽

2009 ◽

Vol 52 (3) ◽

pp. 201-207 ◽

Cited By ~ 2

Author(s):

D.R. Kent ◽

W.L. Cody ◽

A.M. Doherty

Keyword(s):

Asymmetric Synthesis ◽

Enzyme Inhibitors ◽

Arginine Mimetics ◽

Derivatives Of

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Design, Synthesis, and Evaluation of AcyclicC-Nucleoside andN-Methylated Derivatives of the Ribitylaminopyrimidine Substrate of Lumazine Synthase as Potential Enzyme Inhibitors and Mechanistic Probes

The Journal of Organic Chemistry ◽

10.1021/jo048975f ◽

2004 ◽

Vol 69 (21) ◽

pp. 6996-7003 ◽

Cited By ~ 18

Author(s):

Jinhua Chen ◽

Thota Sambaiah ◽

Boris Illarionov ◽

Markus Fischer ◽

Adelbert Bacher ◽

...

Keyword(s):

Enzyme Inhibitors ◽

Design Synthesis ◽

Lumazine Synthase ◽

Derivatives Of

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Irreversible enzyme inhibitors. LXXXIX. candidate active-site-directed irreversible inhibitors of dihydrofolic reductase. X. derivatives of 2-amino-5-benzamidopropyl-4-pyrimidinol

Journal of Heterocyclic Chemistry ◽

10.1002/jhet.5570040205 ◽

1967 ◽

Vol 4 (2) ◽

pp. 188-194 ◽

Cited By ~ 1

Author(s):

B. R. Baker ◽

James K. Coward

Keyword(s):

Active Site ◽

Enzyme Inhibitors ◽

Irreversible Inhibitors ◽

Derivatives Of

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Synthesis of 4-deoxy and 4-deoxy-4-halogeno derivatives of l-fucose as potential enzyme inhibitors

Carbohydrate Research ◽

10.1016/0008-6215(91)80150-l ◽

1991 ◽

Vol 209 ◽

pp. 119-129 ◽

Cited By ~ 24

Author(s):

Thisbe K. Lindhorst ◽

Joachim Thiem

Keyword(s):

Enzyme Inhibitors ◽

Derivatives Of

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β-Lactam Derivatives as Enzyme Inhibitors: Carboxy Peptidyl Derivatives of (S)-4-Oxoazetidine-2-carboxylate as Peptidomimetics

Archiv der Pharmazie ◽

10.1002/1521-4184(200105)334:5<167::aid-ardp167>3.0.co;2-o ◽

2001 ◽

Vol 334 (5) ◽

pp. 167-172 ◽

Cited By ~ 7

Author(s):

Martin Schneider ◽

Hans-Hartwig Otto

Keyword(s):

Enzyme Inhibitors ◽

Derivatives Of

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Irreversible enzyme inhibitors. CLXV. Proteolytic enzymes. 15. Inhibition of guinea pig complement by derivatives of m-phenoxypropoxybenzamidine

Journal of Medicinal Chemistry ◽

10.1021/jm00306a020 ◽

1969 ◽

Vol 12 (6) ◽

pp. 1053-1056 ◽

Cited By ~ 6

Author(s):

Bernard Randall Baker ◽

Michael Cory

Keyword(s):

Guinea Pig ◽

Enzyme Inhibitors ◽

Proteolytic Enzymes ◽

Derivatives Of

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