Regioselective One-pot Synthesis of New Unsymmetric Spiro Dihydrofurans in the Reaction of Mixed Two Different Cyclic β-Dicarbonyl Compounds with BrCN and Aldehydes in the Presence of Et3N

2015 ◽  
Vol 62 (3) ◽  
pp. 234-242 ◽  
Author(s):  
Nader Noroozi Pesyan ◽  
Alireza Shokr ◽  
Ali Gharib ◽  
Tuncay Tunç ◽  
Ertan Sahin
Keyword(s):  
One Pot ◽  
Dicarbonyl Compounds ◽  
One Pot Synthesis

The One-Pot Synthesis of Pyridine Derivatives from The Corresponding 1,5-Dicarbonyl Compounds

Heterocycles ◽  
2019 ◽  
Vol 98 (10) ◽  
pp. 1375
Author(s):  
Hiroyuki Konno ◽  
Takeru Miyakoshi ◽  
Hiromichi Mihara ◽  
Yui Kikuchi
Keyword(s):  
Pyridine Derivatives ◽  
One Pot ◽  
Dicarbonyl Compounds ◽  
One Pot Synthesis ◽  
The One

One-Pot Synthesis of 2-Vinylimidazole Derivatives by Reaction of α-Hydroxyimino-β-dicarbonyl Compounds with Allylamine

Synthesis ◽  
1985 ◽  
Vol 1985 (03) ◽  
pp. 300-302 ◽  
Author(s):  
A. C. Veronese ◽  
G. Vecchiati ◽  
S. Sferra ◽  
P. Orlandini
Keyword(s):  
One Pot ◽  
Dicarbonyl Compounds ◽  
One Pot Synthesis

scholarly journals One Pot Synthesis of Micromolar BACE-1 Inhibitors Based on the Dihydropyrimidinone Scaffold and Their Thia and Imino Analogues

Molecules ◽  
2020 ◽  
Vol 25 (18) ◽  
pp. 4152
Author(s):  
Jessica Bais ◽  
Fabio Benedetti ◽  
Federico Berti ◽  
Iole Cerminara ◽  
Sara Drioli ◽  
...  
Keyword(s):  
Inhibitory Activity ◽  
Biginelli Reaction ◽  
Guanidine Hydrochloride ◽  
One Pot ◽  
Dicarbonyl Compounds ◽  
One Pot Synthesis ◽  
Bace 1

A library of dihydropyrimidinones was synthesized via a “one-pot” three component Biginelli reaction using different aldehydes in combination with β-dicarbonyl compounds and urea. Selected 2-thiooxo and 2-imino analogs were also obtained with the Biginelli reaction from thiourea and guanidine hydrochloride, respectively. The products were screened in vitro for their β-secretase inhibitory activity. The majority of the compounds resulted to be active, with IC50 in the range 100 nM–50 μM.

B2(OH)4-mediated one-pot synthesis of tetrahydroquinoxalines from 2-amino(nitro)anilines and 1,2-dicarbonyl compounds in water

2017 ◽  
Vol 4 (11) ◽  
pp. 2175-2178 ◽  
Author(s):  
Sensheng Liu ◽  
Yanmei Zhou ◽  
Yuebo Sui ◽  
Huan Liu ◽  
Haifeng Zhou
Keyword(s):  
Hydrogen Donor ◽  
One Pot ◽  
Dicarbonyl Compounds ◽  
Metal Free ◽  
One Pot Synthesis

A practical one-pot synthesis of tetrahydroquinoxalines from readily available 2-amino(nitro)anilines and 1,2-dicarbonyl compounds mediated by diboronic acid with water as both a solvent and a hydrogen donor under metal-free conditions has been discovered.

A Facile and Convenient One-Pot Synthesis of Polysubstituted Thiophenes from 1,3-Dicarbonyl Compounds in Water.

ChemInform ◽  
2007 ◽  
Vol 38 (27) ◽  
Author(s):  
Yan Wang ◽  
Dewen Dong ◽  
Yang Yang ◽  
Jie Huang ◽  
Yan Ouyang ◽  
...  
Keyword(s):  
One Pot ◽  
Dicarbonyl Compounds ◽  
One Pot Synthesis
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