Allosteric modulation of the rat adenosine A1 receptor: Differential effects on agonist and antagonist binding

10.1002/ddr.1 ◽  
2000 ◽  
Vol 51 (4) ◽  
pp. 207-215 ◽  
Author(s):  
Angeliki P. Kourounakis ◽  
Corine Visser ◽  
Miriam de Groote ◽  
Ad P. IJzerman
Keyword(s):  
Allosteric Modulation ◽  
Adenosine A1 Receptor ◽  
Differential Effects ◽  
Adenosine A1 ◽  
Agonist And Antagonist ◽  
A1 Receptor ◽  
Antagonist Binding

Differential effects of adenosine A1 receptor on pain-related behavior in normal and nerve-injured rats

2010 ◽  
Vol 1361 ◽  
pp. 23-30 ◽  
Author(s):  
Qing-Juan Gong ◽  
Yu-Ying Li ◽  
Wen-Jun Xin ◽  
Xu-Hong Wei ◽  
Yue Cui ◽  
...  
Keyword(s):  
Adenosine A1 Receptor ◽  
Differential Effects ◽  
Adenosine A1 ◽  
A1 Receptor

The role of the second and third extracellular loops of the adenosine A1 receptor in activation and allosteric modulation

2012 ◽  
Vol 84 (1) ◽  
pp. 76-87 ◽  
Author(s):  
M.C. Peeters ◽  
L.E. Wisse ◽  
A. Dinaj ◽  
B. Vroling ◽  
G. Vriend ◽  
...  
Keyword(s):  
Allosteric Modulation ◽  
Adenosine A1 Receptor ◽  
Extracellular Loops ◽  
Adenosine A1 ◽  
A1 Receptor

A model for the antagonist binding site on the adenosine A1 receptor, based on steric, electrostatic, and hydrophobic properties

1990 ◽  
Vol 33 (6) ◽  
pp. 1708-1713 ◽  
Author(s):  
Philip J. M. Van Galen ◽  
Herman W. T. Van Vlijmen ◽  
Adriaan P. IJzerman ◽  
Willem Soudijn
Keyword(s):  
Binding Site ◽  
Adenosine A1 Receptor ◽  
Hydrophobic Properties ◽  
Adenosine A1 ◽  
A1 Receptor ◽  
Antagonist Binding

scholarly journals Chronic adenosine A1 receptor agonist and antagonist: effect on receptor density and induced seizures in mice

1994 ◽  
Vol 253 (1-2) ◽  
pp. 95-99 ◽  
Author(s):  
Dag K.J.E. Von Lubitz ◽  
Ian A. Paul ◽  
Xiao-duo Ji ◽  
Margaret Carter ◽  
Kenneth A. Jacobson
Keyword(s):  
Receptor Agonist ◽  
Adenosine A1 Receptor ◽  
Receptor Density ◽  
Adenosine A1 ◽  
Agonist And Antagonist ◽  
A1 Receptor ◽  
Antagonist Effect

Repeated treatment with adenosine A1 receptor agonist and antagonist modifies the anticonvulsant properties of CPPene

1996 ◽  
Vol 317 (2-3) ◽  
pp. 239-245 ◽  
Author(s):  
Giovambattista De Sarro ◽  
Eugenio Donato Di Paola ◽  
Umberto Falconi ◽  
Guido Ferreri ◽  
Angela De Sarro
Keyword(s):  
Receptor Agonist ◽  
Adenosine A1 Receptor ◽  
Repeated Treatment ◽  
Adenosine A1 ◽  
Agonist And Antagonist ◽  
A1 Receptor

scholarly journals Allosteric modulation of adenosine A1 receptor coupling to G-proteins in brain

2005 ◽  
Vol 93 (3) ◽  
pp. 715-723 ◽  
Author(s):  
Steven R. Childers ◽  
Xinhui Li ◽  
Ruoyu Xiao ◽  
James C. Eisenach
Keyword(s):  
G Proteins ◽  
Allosteric Modulation ◽  
Adenosine A1 Receptor ◽  
Receptor Coupling ◽  
Adenosine A1 ◽  
A1 Receptor
Sign in / Sign up

Export Citation Format

Share Document