ChemInform Abstract: Design, Synthesis and Characterization of New 1,2,3-Triazolyl Pyrazole Derivatives as Potential Antimicrobial Agents via a Vilsmeier-Haack Reaction Approach.

ChemInform ◽  
2016 ◽  
Vol 47 (45) ◽  
Author(s):  
Manjunatha Bhat ◽  
G. K. Nagaraja ◽  
Reshma Kayarmar ◽  
S. K. Peethamber ◽  
R. Mohammed Shafeeulla
Keyword(s):  
Antimicrobial Agents ◽  
Synthesis And Characterization ◽  
Pyrazole Derivatives ◽  
Design Synthesis

Design, synthesis and characterization of new 1,2,3-triazolyl pyrazole derivatives as potential antimicrobial agents via a Vilsmeier–Haack reaction approach

RSC Advances ◽  
2016 ◽  
Vol 6 (64) ◽  
pp. 59375-59388 ◽  
Author(s):  
Manjunatha Bhat ◽  
Nagaraja G. K. ◽  
Reshma Kayarmar ◽  
Peethamber S. K. ◽  
Mohammed Shafeeulla R
Keyword(s):  
Antimicrobial Agents ◽  
Synthesis And Characterization ◽  
Pyrazole Derivatives ◽  
Design Synthesis ◽  
Anti Oxidant ◽  
Anti Fungal

A new series of 1,2,3-triazolyl pyrazole derivatives were synthesisedviaa Vilsmeier–Haack reaction approach and screened for theirin vitroanti-bacterial, anti-fungal and anti-oxidant activities.

Design, synthesis and characterization of peptidyl boronate analogues as effective antimicrobial agents

2017 ◽  
Vol 43 (10) ◽  
pp. 5755-5778 ◽  
Author(s):  
D. V. R. Venugopal ◽  
Amperayani Karteek Rao ◽  
Parimi Uma Devi ◽  
Y. N. Sastry ◽  
K. Aruna Lakshmi ◽  
...  
Keyword(s):  
Antimicrobial Agents ◽  
Synthesis And Characterization ◽  
Design Synthesis

Design, synthesis, and characterization of novel pyrimidines bearing indole as antimicrobial agents

2018 ◽  
Vol 66 (2) ◽  
pp. 218-225 ◽  
Author(s):  
Mostafa Sayed ◽  
Adel M. Kamal El-Dean ◽  
Mostafa Ahmed ◽  
Reda Hassanien
Keyword(s):  
Antimicrobial Agents ◽  
Synthesis And Characterization ◽  
Design Synthesis

Design, synthesis and characterization of functionalized pyrazole derivatives bearing amide and sulfonamide moieties from aza-aurones

2020 ◽  
Vol 132 (1) ◽  
Author(s):  
Mohammed Chalkha ◽  
Mohamed Bakhouch ◽  
Mohamed Akhazzane ◽  
Mohamed Bourass ◽  
Yohann Nicolas ◽  
...  
Keyword(s):  
Synthesis And Characterization ◽  
Pyrazole Derivatives ◽  
Design Synthesis

scholarly journals Design of an n-type low glass transition temperature radical polymer

2021 ◽  
Author(s):  
Teng Chi ◽  
Siddhartha Akkiraju ◽  
Zihao Liang ◽  
Ying Tan ◽  
Ho Joong Kim ◽  
...  
Keyword(s):  
Glass Transition ◽  
Transition Temperature ◽  
Glass Transition Temperature ◽  
Synthesis And Characterization ◽  
Design Synthesis

We document the design, synthesis, and characterization of the first low glass transition temperature, n-type (i.e., preferentially-reduced) radical polymer.

scholarly journals Novel Acetohydrazide Pyrazole Derivatives: Design, Synthesis, Characterization and Antimicrobial Activity

2019 ◽  
Vol 31 (12) ◽  
pp. 2740-2744
Author(s):  
Anil Verma ◽  
Vinod Kumar ◽  
Ramesh Kataria ◽  
Joginder Singh
Keyword(s):  
Mass Spectrometry ◽  
Antimicrobial Activity ◽  
Antimicrobial Agents ◽  
Antimicrobial Activities ◽  
Pyrazole Derivatives ◽  
Reaction Conditions ◽  
Design Synthesis ◽  
Structure Activity ◽  
Electron Withdrawing Group ◽  
Sar Study

Eleven acetohydrazide linked pyrazole derivatives were designed and synthesized via condensation of acetohyadrazide with different substituted formyl pyrazole derivatives under mild reaction conditions. Synthesized compounds were characterized on the basis of IR, NMR (1H & 13C) and mass spectrometry. The antimicrobial activities of all the compounds were screened against four bacterial and two fungal strains. Among the synthesized compounds, three compounds viz. 6b, 6c and 6d were found as efficient antimicrobial agents in reference to the standard drugs viz. ciprofloxacin and amphotericin-B. Further, structure-activity relationship (SAR) study revealed that electron-withdrawing group enhances the antimicrobial potential of synthesized derivatives as compared to other groups present in the ring. Hence, among compounds 6b-c, compound 6d could be explored further against other microbes to prove its vitality.

Design, Synthesis, and Characterization of Novel CXCR4 Antagonists Featuring Cyclic Amines

ChemMedChem ◽  
2020 ◽  
Vol 15 (13) ◽  
pp. 1150-1162
Author(s):  
Yu Lin ◽  
Zhanhui Li ◽  
Haikuo Ma ◽  
Yujie Wang ◽  
Xu Wang ◽  
...  
Keyword(s):  
Synthesis And Characterization ◽  
Design Synthesis ◽  
Cyclic Amines ◽  
Cxcr4 Antagonists
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