ChemInform Abstract: Overview of Structure, Properties and Derivatives of Boronic Acid

ChemInform ◽  
2015 ◽  
Vol 46 (10) ◽  
pp. no-no
Author(s):  
Aastha Pareek ◽  
Priyanka Rani ◽  
Navneet Kumar ◽  
Pratima Sharma ◽  
D. Kishore
Keyword(s):  
Boronic Acid ◽  
Derivatives Of ◽  
Structure Properties

scholarly journals Synthesis, Complex Compounds and Antimicrobial Activity of Some Derivatives of Furo[3,2-C]Pyridine and Their Starting Compounds

2012 ◽  
Vol 11 (1) ◽  
pp. 73-85
Author(s):  
Martin Hrašna ◽  
Eva Ürgeová ◽  
Alžbeta Krutošíková
Keyword(s):  
Antimicrobial Activity ◽  
Boronic Acid ◽  
Erwinia Amylovora ◽  
Phosphorus Oxychloride ◽  
Coupling Reaction ◽  
Complex Compounds ◽  
Suzuki Coupling Reaction ◽  
Propenoic Acid ◽  
Unexpected Product ◽  
Derivatives Of

Synthesis, Complex Compounds and Antimicrobial Activity of Some Derivatives of Furo[3,2-C]Pyridine and Their Starting CompoundsSome [3,2-c]pyridine derivatives were synthesized. 3-(Furan-2-yl)propenoic acid (1a) was prepared from furan-2-carbaldehyde under the Perkin's conditions. Obtained acid was converted to the corresponding azide3, which in turn was cyclized to give furo[3,2-c]pyridin-4(5H)-one (4a). The reaction of pyridone4awith phosphorus oxychloride rendered the chloroderivative7a, which was treated in the condition of Suzuki coupling reaction with boronic acid to give 4-phenylfuro[3,2-c]pyridine (8e) and an unexpected product10. Some title compounds have shown moderate to good antimicrobial activity against tested bacteriaXanthomonas sp., Erwinia amylovora, and filamentous fungiPyrenophora avenae, Fusarium graminearum.

Novel boronic acid derivatives of bis(indolyl) methane as anti-MRSA agents

2017 ◽  
Vol 27 (10) ◽  
pp. 2135-2138 ◽  
Author(s):  
Santi M. Mandal ◽  
Rupa Pegu ◽  
William F. Porto ◽  
Octavio L. Franco ◽  
Sanjay Pratihar
Keyword(s):  
Boronic Acid ◽  
Boronic Acid Derivatives ◽  
Derivatives Of

Structure–activity relationship of boronic acid derivatives of tyropeptin: Proteasome inhibitors

2010 ◽  
Vol 20 (19) ◽  
pp. 5839-5842 ◽  
Author(s):  
Takumi Watanabe ◽  
Hikaru Abe ◽  
Isao Momose ◽  
Yoshikazu Takahashi ◽  
Daishiro Ikeda ◽  
...  
Keyword(s):  
Boronic Acid ◽  
Proteasome Inhibitors ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Boronic Acid Derivatives ◽  
Relationship Of ◽  
Derivatives Of

Structure Properties Relationship of Donor–Acceptor Derivatives of Triphenylamine and 1,8-Naphthalimide

2012 ◽  
Vol 116 (28) ◽  
pp. 14811-14819 ◽  
Author(s):  
Dalius Gudeika ◽  
Asta Michaleviciute ◽  
Juozas V. Grazulevicius ◽  
Ramunas Lygaitis ◽  
Saulius Grigalevicius ◽  
...  
Keyword(s):  
Donor Acceptor ◽  
Relationship Of ◽  
Derivatives Of ◽  
Structure Properties

scholarly journals 2,4-STUD 2,4-STUDY OF THE STRUC Y OF THE STRUCTURE OF THE P TURE OF THE PAIR EXCHANGE DERIVATIVES E TIVES ETHYL ESTER DIO YL ESTER DIOXOPENTANOATE ACID BY THE METHOD OF PMR AND SAR

2020 ◽  
Vol 4 (2) ◽  
pp. 3-8
Author(s):  
Bako Bafoevich Umarov ◽  
◽  
Murod Amonovich Tursunov ◽  
Mansur Yarashovich Ergashov
Keyword(s):  
Language Learning ◽  
Second Language Learning ◽  
Complex Structure ◽  
Complex Molecules ◽  
Pair Exchange ◽  
Composition Structure ◽  
Relationship Of ◽  
Derivatives Of ◽  
Structure Properties

Analysis of the scientific literature shows that data on nitrogenous derivatives of ketoaldehyde and ketoesters, their synthesis, tautomerization and Complexing ability are incomplete, in some cases their coordination compounds remain abstract, which requires special attention. As a result of the study of the electronic and spatial structures of the complex molecules, it became possible to determine the causes of the "composition-structure-properties" relationship of chemical compounds in a much more complex structure. The structure and tautomerization of para-exchange acylgases of ethyl ether of 2,4-dioxopentanoic acid in various solvents are studied in the article. role of Stephen Krashen's ideas in the theory of second language learning

scholarly journals Novel Boronate Probe Based on 3-Benzothiazol-2-yl-7-hydroxy-chromen-2-one for the Detection of Peroxynitrite and Hypochlorite

Molecules ◽  
2021 ◽  
Vol 26 (19) ◽  
pp. 5940
Author(s):  
Julia Modrzejewska ◽  
Marcin Szala ◽  
Aleksandra Grzelakowska ◽  
Małgorzata Zakłos-Szyda ◽  
Jacek Zielonka ◽  
...  
Keyword(s):  
Fluorescent Probe ◽  
Boronic Acid ◽  
Fast Response ◽  
Fluorescent Detection ◽  
Subsequent Reaction ◽  
Specific Product ◽  
Prolonged Incubation ◽  
Fluorescence Measurements ◽  
Derivatives Of

Derivatives of coumarin, containing oxidant-sensitive boronate group, were recently developed for fluorescent detection of inflammatory oxidants. Here, we report the synthesis and the characterization of 3-(2-benzothiazolyl)-7-coumarin boronic acid pinacol ester (BC-BE) as a fluorescent probe for the detection of peroxynitrite (ONOO–), with high stability and a fast response time. The BC-BE probe hydrolyzes in phosphate buffer to 3-(2-benzothiazolyl)-7-coumarin boronic acid (BC-BA) which is stable in the solution even after a prolonged incubation time (24 h). BC-BA is slowly oxidized by H2O2 to form the phenolic product, 3-benzothiazol-2-yl-7-hydroxy-chromen-2-one (BC-OH). On the other hand, the BC-BA probe reacts rapidly with ONOO−. The ability of the BC-BA probe to detect ONOO– was measured using both authentic ONOO– and the system co-generating steady-state fluxes of O2•– and •NO. BC-BA is oxidized by ONOO– to BC-OH. However, in this reaction 3-benzothiazol-2-yl-chromen-2-one (BC-H) is formed in the minor pathway, as a peroxynitrite-specific product. BC-OH is also formed in the reaction of BC-BA with HOCl, and subsequent reaction of BC-OH with HOCl leads to the formation of a chlorinated phenolic product, which could be used as a specific product for HOCl. We conclude that BC-BA shows potential as an improved fluorescent probe for the detection of peroxynitrite and hypochlorite in biological settings. Complementation of the fluorescence measurements by HPLC-based identification of oxidant-specific products will help to identify the oxidants detected.

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