ChemInform Abstract: Design, Synthesis, and Structureâ€”Activity Relationship of Novel Orally Efficacious Pyrazole/Sulfonamide Based Dihydroquinoline Î³-Secretase Inhibitors.

Gary D. Probst; et al. et al.

doi:10.1002/chin.201003214

ChemInform Abstract: Design, Synthesis, and StructureâActivity Relationship of Novel Orally Efficacious Pyrazole/Sulfonamide Based Dihydroquinoline Î³-Secretase Inhibitors.

ChemInform ◽

10.1002/chin.201003214 ◽

2010 ◽

Vol 41 (3) ◽

Author(s):

Gary D. Probst ◽

et al. et al.

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Relationship Of

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Design, synthesis and structure–activity relationship of simple bis-amides as potent inhibitors of GlyT1

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2008.09.005 ◽

2008 ◽

Vol 18 (20) ◽

pp. 5533-5536 ◽

Cited By ~ 11

Author(s):

Synèse Jolidon ◽

Daniela Alberati ◽

Adam Dowle ◽

Holger Fischer ◽

Dominik Hainzl ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Of

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Design, synthesis, and structure–activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline γ-secretase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2009.07.092 ◽

2009 ◽

Vol 19 (17) ◽

pp. 4920-4923 ◽

Cited By ~ 32

Author(s):

Anh P. Truong ◽

Danielle L. Aubele ◽

Gary D. Probst ◽

Martin L. Neitzel ◽

Chris M. Semko ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Of

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ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationship of Novel Dinucleotide Analogues as Agents Against Herpes and Human Immunodeficiency Viruses.

ChemInform ◽

10.1002/chin.199611278 ◽

2010 ◽

Vol 27 (11) ◽

pp. no-no

Author(s):

G. H. HAKIMELAHI ◽

A. A. MOOSAVI-MOVAHEDI ◽

M. M. SADEGHI ◽

S.-C. TSAY ◽

J. R. HWU

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Human Immunodeficiency Viruses ◽

Relationship Of

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Design, Synthesis, and Structure–Activity Relationship of New Pyrimidinamine Derivatives Containing an Aryloxy Pyridine Moiety

Journal of Agricultural and Food Chemistry ◽

10.1021/acs.jafc.6b05580 ◽

2017 ◽

Vol 65 (6) ◽

pp. 1272-1280 ◽

Cited By ~ 18

Author(s):

Aiying Guan ◽

Changling Liu ◽

Wei Chen ◽

Fan Yang ◽

Yong Xie ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Pyridine Moiety ◽

Structure Activity ◽

Relationship Of

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Design, synthesis and structure–activity relationship of N-substituted tropane muscarinic acetylcholine receptor antagonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.02.015 ◽

2012 ◽

Vol 22 (9) ◽

pp. 3366-3369 ◽

Cited By ~ 3

Author(s):

Dramane I. Lainé ◽

Hongxing Yan ◽

Haibo Xie ◽

Roderick S. Davis ◽

Jeremy Dufour ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Muscarinic Acetylcholine Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Receptor Antagonists ◽

Design Synthesis ◽

Muscarinic Acetylcholine ◽

Structure Activity ◽

Relationship Of

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Design, synthesis and structure–activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.07.049 ◽

2013 ◽

Vol 69 ◽

pp. 115-124 ◽

Cited By ~ 21

Author(s):

Shadia A. Galal ◽

Ahmed S. Abdelsamie ◽

Salwa M. Soliman ◽

Jeremie Mortier ◽

Gerhard Wolber ◽

...

Keyword(s):

Tyrosine Kinase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Tyrosine Kinase Receptor ◽

Design Synthesis ◽

Chemopreventive Agent ◽

Structure Activity ◽

Quinoxaline Derivatives ◽

Relationship Of

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Triple reuptake inhibitors: Design, synthesis and structure–activity relationship of benzylpiperidine–tetrazoles

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.07.046 ◽

2017 ◽

Vol 25 (20) ◽

pp. 5278-5289 ◽

Cited By ~ 8

Author(s):

Suresh Paudel ◽

Xiao Min ◽

Srijan Acharya ◽

Daulat Bikram Khadka ◽

Goo Yoon ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Of

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Design, synthesis, and structure–activity relationship of carbamate-tethered aryl propanoic acids as novel PPARα/γ dual agonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.04.057 ◽

2007 ◽

Vol 17 (13) ◽

pp. 3595-3598 ◽

Cited By ~ 13

Author(s):

Nam-Jung Kim ◽

Kwang-Ok Lee ◽

Bon-Woong Koo ◽

Funan Li ◽

Ja-Kyung Yoo ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Of

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Design, synthesis and structure–activity relationship of novel semi-synthetic flavonoids as antiproliferative agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.06.007 ◽

2014 ◽

Vol 82 ◽

pp. 506-520 ◽

Cited By ~ 23

Author(s):

F.A. Ragab ◽

T.A.A. Yahya ◽

M.M. El-Naa ◽

R.K. Arafa

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Antiproliferative Agents ◽

Structure Activity ◽

Relationship Of

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Design, synthesis and the structure-activity relationship of agonists targeting on the ALDH2 catalytic tunnel

Bioorganic Chemistry ◽

10.1016/j.bioorg.2020.104166 ◽

2020 ◽

Vol 104 ◽

pp. 104166

Author(s):

Ming-Che Cheng ◽

Wei-Chi Lo ◽

Yu-Wen Chang ◽

Shoei-Sheng Lee ◽

Chia-Chuan Chang

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Of

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ChemInform Abstract: Design, Synthesis, and StructureâActivity Relationship of Novel Orally Efficacious Pyrazole/Sulfonamide Based Dihydroquinoline Î³-Secretase Inhibitors.

Design, synthesis and structure–activity relationship of simple bis-amides as potent inhibitors of GlyT1

Design, synthesis, and structure–activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline γ-secretase inhibitors

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationship of Novel Dinucleotide Analogues as Agents Against Herpes and Human Immunodeficiency Viruses.

Design, Synthesis, and Structure–Activity Relationship of New Pyrimidinamine Derivatives Containing an Aryloxy Pyridine Moiety

Design, synthesis and structure–activity relationship of N-substituted tropane muscarinic acetylcholine receptor antagonists

Design, synthesis and structure–activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor

Triple reuptake inhibitors: Design, synthesis and structure–activity relationship of benzylpiperidine–tetrazoles

Design, synthesis, and structure–activity relationship of carbamate-tethered aryl propanoic acids as novel PPARα/γ dual agonists

Design, synthesis and structure–activity relationship of novel semi-synthetic flavonoids as antiproliferative agents

Design, synthesis and the structure-activity relationship of agonists targeting on the ALDH2 catalytic tunnel

ChemInform Abstract: Design, Synthesis, and StructureâActivity Relationship of Novel Orally Efficacious Pyrazole/Sulfonamide Based Dihydroquinoline Î³-Secretase Inhibitors.