ChemInform Abstract: Facile Synthesis of Benzo[4,5]furo[3,2-c]pyridines via Palladium-catalyzed Intramolecular Heck Reaction.

ChemInform ◽  
2009 ◽  
Vol 40 (46) ◽  
Author(s):  
Woo Sub Yoon ◽  
Su Jung Lee ◽  
Seung Kyu Kang ◽  
Deok-Chan Ha ◽  
Jae Du Ha
Keyword(s):  
Heck Reaction ◽  
Facile Synthesis ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

Facile synthesis of benzo[4,5]furo[3,2-c]pyridines via palladium-catalyzed intramolecular Heck reaction

2009 ◽  
Vol 50 (31) ◽  
pp. 4492-4494 ◽  
Author(s):  
Woo Sub Yoon ◽  
Su Jung Lee ◽  
Seung Kyu Kang ◽  
Deok-Chan Ha ◽  
Jae Du Ha
Keyword(s):  
Heck Reaction ◽  
Facile Synthesis ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

Ligand promoted and controlled palladium-catalyzed intramolecular Heck reaction of homoallyl alcohols: a facile synthesis of cyclopentaannulated quinolines

Tetrahedron ◽  
2012 ◽  
Vol 68 (45) ◽  
pp. 9206-9210 ◽  
Author(s):  
Radhey M. Singh ◽  
Atish Chandra ◽  
Neha Sharma ◽  
Bhawana Singh ◽  
Ritush Kumar
Keyword(s):  
Heck Reaction ◽  
Facile Synthesis ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

Palladium-Catalyzed 8-Exo Trig Intramolecular Heck Reaction Under Microwave Irradiation in the Presence of Basic Alumina

2012 ◽  
Vol 42 (21) ◽  
pp. 3166-3176 ◽  
Author(s):  
Pritam Saha ◽  
Shyamal Mondal ◽  
Abhijit Hazra ◽  
Subhendu Naskar ◽  
Arindam Maity ◽  
...  
Keyword(s):  
Microwave Irradiation ◽  
Heck Reaction ◽  
Basic Alumina ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

ChemInform Abstract: Ligand-Free Palladium-Catalyzed Intramolecular Heck Reaction of Secondary Benzylic Bromides.

ChemInform ◽  
2011 ◽  
Vol 42 (52) ◽  
pp. no-no
Author(s):  
Wei Zhou ◽  
Guanghui An ◽  
Guangqian Zhang ◽  
Jianlin Han ◽  
Yi Pan
Keyword(s):  
Heck Reaction ◽  
Ligand Free ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

Dibenzo[b,e]azepin-6-ones and Seven-Membered Sultam Derivatives: Convenient Synthesis via Palladium-Catalyzed Regioselective Intra­molecular Heck Reaction and Application towards Drug-Like Small Molecules

Synthesis ◽  
2019 ◽  
Vol 51 (17) ◽  
pp. 3231-3240 ◽  
Author(s):  
Arijit Das ◽  
Arup Maiti ◽  
Mrinalkanti Kundu ◽  
Kuldeep K. Roy ◽  
Inul Ansary
Keyword(s):  
Small Molecules ◽  
Acetylcholine Receptor ◽  
Heck Reaction ◽  
Good Yield ◽  
Muscarinic Acetylcholine Receptor ◽  
Binding Potential ◽  
Modeling Studies ◽  
Convenient Synthesis ◽  
Palladium Catalyzed ◽  
Intramolecular Heck Reaction

A new, convenient synthesis of dibenzo[b,e]azepin-6-ones and seven-membered sultam derivatives have been envisaged via Pd-catalyzed regioselective intramolecular Heck reaction of the corresponding easily accessible precursors. This protocol has been successfully implemented to synthesize N-methyldarenzepine in four steps and in good yield. Moreover, one of the intermediates has been utilized for the synthesis of a new analogue of darenzepine. Preliminary modeling studies were performed to investigate the binding potential to muscarinic acetylcholine receptor (M4).

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