ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationship Studies of ATP Analogues as DNA Gyrase Inhibitors.

Thomas Luebbers; Peter Angehrn; Hans Gmuender; Silvia Herzig; Josef Kulhanek

doi:10.1002/chin.200030134

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationship Studies of ATP Analogues as DNA Gyrase Inhibitors.

ChemInform ◽

10.1002/chin.200030134 ◽

2010 ◽

Vol 31 (30) ◽

pp. no-no

Author(s):

Thomas Luebbers ◽

Peter Angehrn ◽

Hans Gmuender ◽

Silvia Herzig ◽

Josef Kulhanek

Keyword(s):

Dna Gyrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Atp Analogues ◽

Gyrase Inhibitors

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Design, synthesis, and structure–activity relationship studies of ATP analogues as DNA gyrase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(00)00109-8 ◽

2000 ◽

Vol 10 (8) ◽

pp. 821-826 ◽

Cited By ~ 61

Author(s):

Thomas Lübbers ◽

Peter Angehrn ◽

Hans Gmünder ◽

Silvia Herzig ◽

Josef Kulhanek

Keyword(s):

Dna Gyrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Atp Analogues ◽

Gyrase Inhibitors

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Design, Synthesis and Structure—Activity Relationship Studies of Novel Indazole Analogues as DNA Gyrase Inhibitors with Gram-Positive Antibacterial Activity.

ChemInform ◽

10.1002/chin.200438127 ◽

2004 ◽

Vol 35 (38) ◽

Author(s):

Akihiko Tanitame ◽

Yoshihiro Oyamada ◽

Keiko Ofuji ◽

Yoko Kyoya ◽

Kenji Suzuki ◽

...

Keyword(s):

Antibacterial Activity ◽

Dna Gyrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Gram Positive ◽

Design Synthesis ◽

Structure Activity ◽

Gyrase Inhibitors

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Design, synthesis, and structure–activity relationship studies of new phenolic DNA gyrase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.12.065 ◽

2007 ◽

Vol 17 (16) ◽

pp. 4708-4714 ◽

Cited By ~ 55

Author(s):

Thomas Lübbers ◽

Peter Angehrn ◽

Hans Gmünder ◽

Silvia Herzig

Keyword(s):

Dna Gyrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Gyrase Inhibitors

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Design, synthesis and structure–activity relationship studies of novel indazole analogues as DNA gyrase inhibitors with Gram-positive antibacterial activity

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.03.044 ◽

2004 ◽

Vol 14 (11) ◽

pp. 2857-2862 ◽

Cited By ~ 53

Author(s):

Akihiko Tanitame ◽

Yoshihiro Oyamada ◽

Keiko Ofuji ◽

Yoko Kyoya ◽

Kenji Suzuki ◽

...

Keyword(s):

Antibacterial Activity ◽

Dna Gyrase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Gram Positive ◽

Design Synthesis ◽

Structure Activity ◽

Gyrase Inhibitors

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Quantitative Structure–Activity Relationship Analysis and Validation of New DNA Gyrase Inhibitors

Pharmaceutical Chemistry Journal ◽

10.1007/s11094-021-02513-x ◽

2022 ◽

Author(s):

S. Bhuvaneswari ◽

V. Bala Aakash ◽

N. Ramalakshmi ◽

S. Arunkumar

Keyword(s):

Dna Gyrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Relationship Analysis ◽

Structure Activity ◽

Gyrase Inhibitors

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Design, Synthesis and Structure-Activity Relationship Studies of Novel 4 (1-adamantyl) Phenyl Analogues as HIF-1α Inhibitors

Medicinal Chemistry ◽

10.2174/1573406412666151109113007 ◽

2016 ◽

Vol 12 (4) ◽

pp. 338-346 ◽

Cited By ~ 2

Author(s):

Yan Xia ◽

Qiong Duan ◽

Bao-Hua Zhao ◽

Dong-Feng Li ◽

Rui-Bin Hou

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity

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Design, synthesis, biological evaluation and structure-activity relationship study of quinazolin-4(3H)-one derivatives as novel USP7 inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113291 ◽

2021 ◽

pp. 113291

Author(s):

Peng Li ◽

Ying Liu ◽

Hua Yang ◽

Hong-Min Liu

Keyword(s):

Structure Activity Relationship ◽

Biological Evaluation ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Study

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New substituted pyrazolones and dipyrazolotriazines as promising tyrosyl-tRNA synthetase and peroxiredoxin-5 inhibitors: Design, synthesis, molecular docking and structure-activity relationship (SAR) analysis

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104704 ◽

2021 ◽

Vol 109 ◽

pp. 104704

Author(s):

Ismail M.M. Othman ◽

Mohamed A.M. Gad-Elkareem ◽

El Hassane Anouar ◽

Kaïss Aouadi ◽

Mejdi Snoussi ◽

...

Keyword(s):

Molecular Docking ◽

Structure Activity Relationship ◽

Trna Synthetase ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Sar Analysis

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Antileishmanial Chalcones: Statistical Design, Synthesis, and Three-Dimensional Quantitative Structure−Activity Relationship Analysis

Journal of Medicinal Chemistry ◽

10.1021/jm980410m ◽

1998 ◽

Vol 41 (24) ◽

pp. 4819-4832 ◽

Cited By ~ 183

Author(s):

Simon Feldbæk Nielsen ◽

Søren Brøgger Christensen ◽

Gabriele Cruciani ◽

Arsalan Kharazmi ◽

Tommy Liljefors

Keyword(s):

Three Dimensional ◽

Statistical Design ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Relationship Analysis ◽

Structure Activity

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Novel Pyrazole-4-acetohydrazide Derivatives Potentially Targeting Fungal Succinate Dehydrogenase: Design, Synthesis, Three-Dimensional Quantitative Structure–Activity Relationship, and Molecular Docking

Journal of Agricultural and Food Chemistry ◽

10.1021/acs.jafc.1c03399 ◽

2021 ◽

Author(s):

Xiaobin Wang ◽

Mengqi Wang ◽

Ling Han ◽

Fei Jin ◽

Jian Jiao ◽

...

Keyword(s):

Molecular Docking ◽

Succinate Dehydrogenase ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Structure Activity

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