ChemInform Abstract: Synthesis and Biological Activity of Some New 1-, 2- and 8-Substituted Dibenzothiophene Amino Acid Derivatives.

1983 ◽  
Vol 14 (13) ◽  
Author(s):  
A. M. EL-NAGGAR ◽  
F. M. S. AHMED ◽  
A. M. ABD EL-SALAM ◽  
S. G. DONIA
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Amino Acid Derivatives

Synthesis and biological activity of some new 3-and 6-substituted coumarin amino acid derivatives. Part I

1981 ◽  
Vol 18 (6) ◽  
pp. 1203-1207 ◽  
Author(s):  
A. M. El-Naggar ◽  
F. S. M. Ahmed ◽  
A. M. Abd El-Salam ◽  
M. A. Radi ◽  
M. S. A. Latif
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Amino Acid Derivatives ◽  
Coumarin Amino Acid

?-Amino ketones ? ?-amino acid derivatives. IV. Aminomethyl derivatives of acetophenones and their biological activity

1984 ◽  
Vol 18 (6) ◽  
pp. 403-409
Author(s):  
A. G. Agababyan ◽  
G. A. Gevorgyan ◽  
L. K. Durgaryan ◽  
�. V. Vlasenko ◽  
R. V. Agababyan ◽  
...  
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Amino Acid Derivatives ◽  
Aminomethyl Derivatives ◽  
Derivatives Of

Synthesis of thiosulphonate and amino acid derivatives of benzochinone and predicted screening of their biological activity

2021 ◽  
Vol 4 (2) ◽  
pp. 40-46
Author(s):  
N. Y. Monka ◽  
◽  
L. R. Zhurakhivska ◽  
M. S. Kurka ◽  
G. B. Shiуan ◽  
...  
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Experimental Studies ◽  
Physicochemical Characteristics ◽  
Biologically Active ◽  
Amino Acid Derivatives ◽  
Online Resource ◽  
Methods Of Synthesis ◽  
Pass Online

Quinoid derivatives are attractive not only as interesting synthons for synthesis, but also as potential biologically active substances, so it is important to modify the compounds of the quinone series with different pharmacoform fragments. In this work, the structural design of chlorine and bromanyl disulfur-containing fragments, namely thiosulfonate, and chloranyl – a fragment of 4- aminobutanoic acid. Methods of synthesis were developed and physicochemical characteristics of thiosulfonate and amino acid derivatives were studied: 2,5-bis (thiosulfonate) -3,6-halogen -1,4- benzoquinones and 2,5-bis (3-carboxypropylamino) -3,6 - dichlorobenzoquinone. The prospects for the design of chlorine and bromanyl thiosulfonate fragments and chloranyl fragment of 4- aminobutanoic acid are confirmed by the results of predicting the biological activity of 5 a, b, 6 a, b, 7 using the online resource PASS Online. In particular, the substance 6a obtained by us is promising in terms of research on Antiviral (Picornavirus). The obtained results of predicted cytotoxicity screening indicate the feasibility of conducting experimental studies by in vitro methods on anticancer activity against cancer cell lines of hematopoietic and lymphoid tissue, lungs, skin, ovaries, blood, breast, kidney, colon, brain.

scholarly journals Antibiotics Aminosidin (Paromomycin). III. Some Amino Acid Derivatives and Their Biological Activity

1976 ◽  
Vol 96 (5) ◽  
pp. 557-564
Author(s):  
YOSUKE SAWADA ◽  
TETSU OKUNO ◽  
HYOZO TANIYAMA
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Amino Acid Derivatives

Synthesis and biological activity of amino acid derivatives of sulfanilic acid

1982 ◽  
Vol 16 (7) ◽  
pp. 520-524
Author(s):  
N. M. Divanyan ◽  
L. Kh. Galstyan ◽  
A. A. Chachoyan ◽  
B. T. Garibdzhanyan ◽  
N. O. Stepanyan ◽  
...  
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Sulfanilic Acid ◽  
Amino Acid Derivatives ◽  
Derivatives Of

Synthesis, Characterization, and Biological Activity of Amino Acid Derivatives of the Heteropolytungstophosphoric Acid

2006 ◽  
Vol 137 (6) ◽  
pp. 803-810 ◽  
Author(s):  
Vesna Kuntić ◽  
Maja Stanojević ◽  
Ivanka Holclajtner-Antunović ◽  
Snežana Uskoković-Marković ◽  
Ubavka Mioč ◽  
...  
Keyword(s):  
Biological Activity ◽  
Amino Acid ◽  
Amino Acid Derivatives ◽  
Derivatives Of
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