Synthesis of Ribo‐Azanucleosides by Anodic Oxidation: Reactivity Control of Intermediate for Efficient Access to Pharmacophores

2018 ◽  
Vol 24 (68) ◽  
pp. 17902-17905 ◽  
Author(s):  
Kazuhiro Okamoto ◽  
Takao Shoji ◽  
Mizuki Tsutsui ◽  
Naoki Shida ◽  
Kazuhiro Chiba
2014 ◽  
Vol 25 (8) ◽  
pp. 1112-1114 ◽  
Author(s):  
Jia-Qian Ye ◽  
Zhen-Lei Zhang ◽  
Zheng-Gen Zha ◽  
Zhi-Yong Wang

ChemInform ◽  
2014 ◽  
Vol 46 (3) ◽  
pp. no-no
Author(s):  
Jia-Qian Ye ◽  
Zhen-Lei Zhang ◽  
Zheng-Gen Zha ◽  
Zhi-Yong Wang

2019 ◽  
Author(s):  
Nicolas Duchemin ◽  
Roberto Buccafusca ◽  
Marc Daumas ◽  
Vincent Ferey ◽  
Stellios Arseniyadis

We report here a general method that allows a highly straightforward access to tertiary difluoromethylated compounds. The strategy relies on a two-step sequence featuring a C-selective electrophilic difluoromethylation and an unprecedented palladium-catalyzed decarboxylative protonation. Considering the generality of the method and the attractive properties offered by the difluoromethyl group, this approach provides a valuable tool for late-stage functionalization and drug development.<br>


Author(s):  
A.S. Kamysheva ◽  
◽  
A.I. Koroleva ◽  
L.P. Mileshko ◽  
◽  
...  

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