A One-PotO-Phosphinative Passerini/Pudovik Reaction: Efficient Synthesis of Highly Functionalized α-(Phosphinyloxy)amide Derivatives

2014 ◽  
Vol 20 (17) ◽  
pp. 5007-5012 ◽  
Author(s):  
Takahiro Soeta ◽  
Syunsuke Matsuzaki ◽  
Yutaka Ukaji
Synthesis ◽  
2017 ◽  
Vol 49 (11) ◽  
pp. 2435-2442 ◽  
Author(s):  
Prashantha Kamath ◽  
Ramya Rajan ◽  
Sudhindra Deshpande ◽  
Mark Montgomery ◽  
Mukul Lal

A simple, fast and efficient synthesis of 3-phosphorylated benzoxaboroles using the Pudovik reaction is reported. A number of diverse 3-(dialkoxyphosphoryl)-1-hydroxy-3H-2,1-benzoxaboroles were synthesised in 70–86% yield. Interesting hydrogen bond features were observed in the crystal lattice of the 5-chlorinated 3-bis(benzyl­oxy)phosphoryl derivative with both inter- and intramolecular C–H···O hydrogen bonds. Additionally, linear chains of intermolecular O–H···O hydrogen bonds were observed.


Planta Medica ◽  
2009 ◽  
Vol 75 (09) ◽  
Author(s):  
LA Vilaseca ◽  
J Quillaguamán ◽  
L Fuentes ◽  
O Sterner
Keyword(s):  

2014 ◽  
Vol 34 (1) ◽  
pp. 243-250
Author(s):  
Jianghong DING ◽  
Le XU ◽  
Hao XU ◽  
Haihong WU ◽  
Yueming LIU ◽  
...  

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