Examples of Peptide-Peptoid Hybrid Serine Protease Inhibitors Based on the Trypsin Inhibitor SFTI-1 with Complete Protease Resistance at the P1P1′ Reactive Site

Maciej Stawikowski; Roma Stawikowska; Anna Jaśkiewicz; Ewa Zabłotna; Krzysztof Rolka

doi:10.1002/cbic.200400412

Examples of Peptide-Peptoid Hybrid Serine Protease Inhibitors Based on the Trypsin Inhibitor SFTI-1 with Complete Protease Resistance at the P1P1′ Reactive Site

ChemBioChem ◽

10.1002/cbic.200400412 ◽

2005 ◽

Vol 6 (6) ◽

pp. 1057-1061 ◽

Cited By ~ 34

Author(s):

Maciej Stawikowski ◽

Roma Stawikowska ◽

Anna Jaśkiewicz ◽

Ewa Zabłotna ◽

Krzysztof Rolka

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Trypsin Inhibitor ◽

Serine Protease Inhibitors ◽

Reactive Site ◽

Protease Resistance

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A New Family of Serine Protease Inhibitors (Bombyx Family) as Established from the Unique Topological Relation between the Positions of Disulfide Bridges and Reactive Site

The Journal of Biochemistry ◽

10.1093/oxfordjournals.jbchem.a021259 ◽

1996 ◽

Vol 119 (3) ◽

pp. 428-434 ◽

Cited By ~ 20

Author(s):

M. Itoh ◽

T.-N. Pham ◽

K. Hayashi ◽

R. Takano ◽

M. Eguchi ◽

...

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Disulfide Bridges ◽

Serine Protease Inhibitors ◽

Reactive Site ◽

Topological Relation ◽

New Family

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Synthesis of a mixture of cyclic peptides based on the Bowman-Birk reactive site loop to screen for serine protease inhibitors

International journal of peptide & protein research ◽

10.1111/j.1399-3011.1995.tb00585.x ◽

2009 ◽

Vol 46 (1) ◽

pp. 79-87 ◽

Cited By ~ 33

Author(s):

GONZALO J. DOMINGO ◽

ROBIN J. LEATHERBARROW ◽

NEIL FREEMAN ◽

SHILA PATEL ◽

MALCOLM WEIR

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Cyclic Peptides ◽

Serine Protease Inhibitors ◽

Reactive Site

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Anisakis simplex:Mutational Bursts in the Reactive Site Centers of Serine Protease Inhibitors from an Ascarid Nematode

Experimental Parasitology ◽

10.1006/expr.1998.4284 ◽

1998 ◽

Vol 89 (2) ◽

pp. 257-261 ◽

Cited By ~ 17

Author(s):

Cheng-Chan Lu ◽

Tien Nguyen ◽

Stephen Morris ◽

Dolores Hill ◽

Judy A. Sakanari

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Serine Protease Inhibitors ◽

Reactive Site

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Effect of serine protease inhibitors on the expression of cell surface and soluble forms of two types of tumor necrosis factor receptors

Immunology Letters ◽

10.1016/s0165-2478(97)87943-6 ◽

1997 ◽

Vol 56 (1-3) ◽

pp. 276

Author(s):

E Pócsik

Keyword(s):

Tumor Necrosis Factor ◽

Cell Surface ◽

Serine Protease ◽

Protease Inhibitors ◽

Tumor Necrosis ◽

Serine Protease Inhibitors ◽

Tumor Necrosis Factor Receptors ◽

Necrosis Factor

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Detection and analysis of hepatitis C virus NS3 serine protease inhibitors

Journal of Hepatology ◽

10.1016/s0168-8278(01)80459-1 ◽

2001 ◽

Vol 34 (0) ◽

pp. 126-127

Author(s):

R Zemel

Keyword(s):

Hepatitis C Virus ◽

Hepatitis C ◽

Serine Protease ◽

Protease Inhibitors ◽

Serine Protease Inhibitors

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Serine protease inhibitors from Amazon leguminosae seeds: purification and preliminary characterization of two chymotrypsin inhibitors from Inga umbratica

Protein and Peptide Letters ◽

10.2174/0929866013409175 ◽

2001 ◽

Vol 8 (6) ◽

pp. 485-493 ◽

Cited By ~ 8

Author(s):

A. Calderon ◽

R. Teles ◽

J.R. Leite ◽

Jr Bloch ◽

S. Astolfi-Filho ◽

...

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Serine Protease Inhibitors ◽

Preliminary Characterization ◽

Chymotrypsin Inhibitors

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Development of Trypsin-Like Serine Protease Inhibitors as Therapeutic Agents: Opportunities, Challenges, and their Unique Structure-Based Rationales

Current Topics in Medicinal Chemistry ◽

10.2174/1568026615666150915121447 ◽

2016 ◽

Vol 16 (13) ◽

pp. 1506-1529 ◽

Cited By ~ 8

Author(s):

Guyan Liang ◽

J. Phillip Bowen

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Therapeutic Agents ◽

Serine Protease Inhibitors ◽

Unique Structure

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A collagen-binding protein in the endoplasmic reticulum of myoblasts exhibits relationship with serine protease inhibitors.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(19)47363-8 ◽

1991 ◽

Vol 266 (26) ◽

pp. 17230-17235 ◽

Cited By ~ 1

Author(s):

E.P. Clarke ◽

G.A. Cates ◽

E.H. Ball ◽

B.D. Sanwal

Keyword(s):

Endoplasmic Reticulum ◽

Serine Protease ◽

Protease Inhibitors ◽

Binding Protein ◽

Serine Protease Inhibitors ◽

Collagen Binding

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Synergistic effect of serine protease inhibitors and a bothropic antivenom in reducing local hemorrhage and coagulopathy caused by Bothrops jararaca venom

Toxicon ◽

10.1016/j.toxicon.2021.06.009 ◽

2021 ◽

Author(s):

G.M. Silva ◽

D.H. Berto ◽

C.A. Lima ◽

K.B. Waitman ◽

C.F.G. Lima ◽

...

Keyword(s):

Synergistic Effect ◽

Serine Protease ◽

Protease Inhibitors ◽

Serine Protease Inhibitors ◽

Bothrops Jararaca

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Calpain Inhibitors and Serine Protease Inhibitors Can Produce Apoptosis in HL-60 Cells

Archives of Biochemistry and Biophysics ◽

10.1006/abbi.1996.0443 ◽

1996 ◽

Vol 334 (1) ◽

pp. 175-181 ◽

Cited By ~ 33

Author(s):

Qin Lu ◽

Ronald L. Mellgren

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Serine Protease Inhibitors ◽

Calpain Inhibitors

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