Monitoring Ligand-Induced Conformational Changes for the Identification of Estrogen Receptor Agonists and Antagonists

Svenja C. Mayer-Wrangowski; Daniel Rauh

doi:10.1002/anie.201410148

Monitoring Ligand-Induced Conformational Changes for the Identification of Estrogen Receptor Agonists and Antagonists

Angewandte Chemie International Edition ◽

10.1002/anie.201410148 ◽

2015 ◽

Vol 54 (14) ◽

pp. 4379-4382 ◽

Cited By ~ 14

Author(s):

Svenja C. Mayer-Wrangowski ◽

Daniel Rauh

Keyword(s):

Estrogen Receptor ◽

Conformational Changes ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists

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Test No. 457: BG1Luc Estrogen Receptor Transactivation Test Method for Identifying Estrogen Receptor Agonists and Antagonists

10.1787/9789264185395-en ◽

2012 ◽

Cited By ~ 7

Author(s):

Keyword(s):

Estrogen Receptor ◽

Test Method ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists ◽

Receptor Transactivation

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Test No. 455: Performance-Based Test Guideline for Stably Transfected Transactivation In Vitro Assays to Detect Estrogen Receptor Agonists and Antagonists

10.1787/9789264243040-en ◽

2015 ◽

Cited By ~ 1

Author(s):

Keyword(s):

Estrogen Receptor ◽

In Vitro Assays ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists ◽

Test Guideline

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Analysis of the molecular pharmacology of estrogen receptor agonists and antagonists provides insights into the mechanism of action of estrogen in bone

Osteoporosis International ◽

10.1007/bf01674810 ◽

1997 ◽

Vol 7 (S1) ◽

pp. 29-34 ◽

Cited By ~ 28

Author(s):

D. P. McDonnell ◽

J. D. Norris

Keyword(s):

Estrogen Receptor ◽

Mechanism Of Action ◽

Molecular Pharmacology ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists

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Human estrogen receptor regulation in a yeast model system and studies on receptor agonists and antagonists

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/0960-0760(92)90108-u ◽

1992 ◽

Vol 42 (7) ◽

pp. 677-685 ◽

Cited By ~ 67

Author(s):

C.Richard Lyttle ◽

P. Damian-Matsumura ◽

H. Juul ◽

Tauseef R. Butt

Keyword(s):

Estrogen Receptor ◽

Model System ◽

Receptor Regulation ◽

Receptor Agonists ◽

Human Estrogen Receptor ◽

Receptor Agonists And Antagonists ◽

Yeast Model

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Failure of Topical Estrogen Receptor Agonists and Antagonists to Alter Murine Hair Follicle Cycling

Journal of Investigative Dermatology ◽

10.1046/j.1523-1747.1998.00077.x ◽

1998 ◽

Vol 110 (1) ◽

pp. 95 ◽

Cited By ~ 5

Author(s):

Kurt S. Stenn ◽

R. Paus ◽

M. Filippi

Keyword(s):

Estrogen Receptor ◽

Hair Follicle ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists ◽

Topical Estrogen

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Modulation of mitochondrial Ca2+ uptake by estrogen receptor agonists and antagonists

British Journal of Pharmacology ◽

10.1038/sj.bjp.0706265 ◽

2005 ◽

Vol 145 (7) ◽

pp. 862-871 ◽

Cited By ~ 34

Author(s):

Carmen D Lobatón ◽

Laura Vay ◽

Esther Hernández-SanMiguel ◽

Jaime SantoDomingo ◽

Alfredo Moreno ◽

...

Keyword(s):

Estrogen Receptor ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists

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Corrigendum to “Synthesis and biological activities of some new dibenzopyranones and dibenzopyrans: search for potential estrogen receptor agonists and antagonists”

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2004.07.001 ◽

2004 ◽

Vol 12 (19) ◽

pp. 5237

Author(s):

Jaya Pandey ◽

Ashok K. Jha ◽

K. Hajela ◽

P.S.N. Murthy ◽

Shikha Sharma ◽

...

Keyword(s):

Estrogen Receptor ◽

Biological Activities ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists

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Test No. 455: Performance-Based Test Guideline for Stably Transfected Transactivation In Vitro Assays to Detect Estrogen Receptor Agonists and Antagonists

10.1787/9789264265295-en ◽

2016 ◽

Cited By ~ 6

Author(s):

Keyword(s):

Estrogen Receptor ◽

In Vitro Assays ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists ◽

Test Guideline

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Combined action of estrogen receptor agonists and antagonists in two-hybrid recombinant yeast in vitro

Ecotoxicology and Environmental Safety ◽

10.1016/j.ecoenv.2014.09.025 ◽

2015 ◽

Vol 111 ◽

pp. 228-235 ◽

Cited By ~ 4

Author(s):

Rong Yang ◽

Na Li ◽

Kaifeng Rao ◽

Mei Ma ◽

Zijian Wang

Keyword(s):

Estrogen Receptor ◽

Recombinant Yeast ◽

Receptor Agonists ◽

Combined Action ◽

Receptor Agonists And Antagonists ◽

Two Hybrid

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Estrogen Receptor Agonists and Antagonists in the Yeast Estrogen Bioassay

Methods in Molecular Biology - Estrogen Receptors ◽

10.1007/978-1-4939-3127-9_26 ◽

2016 ◽

pp. 337-342 ◽

Cited By ~ 2

Author(s):

Si Wang ◽

Toine F. H. Bovee

Keyword(s):

Estrogen Receptor ◽

Receptor Agonists ◽

Receptor Agonists And Antagonists

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