Braces for the Peptide Backbone: Insights into Structure-Activity Relationships of Protease Inhibitor Mimics with Locked Amide Conformations

2012 ◽  
Vol 51 (15) ◽  
pp. 3708-3712 ◽  
Author(s):  
Marco Tischler ◽  
Daichi Nasu ◽  
Martin Empting ◽  
Stefan Schmelz ◽  
Dirk W. Heinz ◽  
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Keyword(s):  
Protease Inhibitor ◽  
Peptide Backbone ◽  
Structure Activity Relationships ◽  
Structure Activity

HIV protease inhibitor HOE/BAY 793, structure-activity relationships in a series of C2-symmetric diols

1995 ◽  
Vol 3 (5) ◽  
pp. 559-571 ◽  
Author(s):  
Karl-Heinz Budt ◽  
Anusch Peyman ◽  
Jutta Hansen ◽  
Jochen Knolle ◽  
Christoph Meichsner ◽  
...  
Keyword(s):  
Protease Inhibitor ◽  
Hiv Protease ◽  
Hiv Protease Inhibitor ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure-activity relationships in the acronycine and benzo[b]acronycine series: Role of the pyran ring

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
Q Do ◽  
H Doan Thi Mai ◽  
T Gaslonde ◽  
B Pfeiffer ◽  
S Léonce ◽  
...  
Keyword(s):  
Pyran Ring ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure activity-relationships of P-Glycoprotein modulation using a small library of macrocyclic lathyrane diterpenes

Planta Medica ◽  
2012 ◽  
Vol 78 (11) ◽  
Author(s):  
M Reis ◽  
RJ Ferreira ◽  
MMM Santos ◽  
DJVA dos Santos ◽  
J Molnár ◽  
...  
Keyword(s):  
Structure Activity Relationships ◽  
Structure Activity ◽  
P Glycoprotein
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